IRIS
GROSSI, GIANCARLO
 Distribuzione geografica
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Continente #
EU - Europa 5.121
Totale 5.121
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Nazione #
IT - Italia 5.121
Totale 5.121
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Città #
Genova 3.657
Genoa 514
Rapallo 507
Vado Ligure 430
Bordighera 13
Totale 5.121
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Nome #
1,2-Fused Pyrimidines. V. Synthesis of 1-Alkyl or Phenyl-2H-dipyrido-[1,2-a:2’, 3’-d]pyrimidine-2,5(1H)-diones 296
1,5-Benzodiazepines IX. A new route to substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines with analgesic and/or anti-inflammatory activities 161
Synthesis, in vitro antiplatelet activity and molecular modelling studies of 10-substituted 2-(1-piperazinyl)pyrimido[1,2-a]benzimidazol-4(10H)-ones 158
1,8-Naphthyridines VIII. Novel 5-aminoimidazo[1,2-a][1,8]naphthyridine-6-carboxamide and 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamide derivatives showing potent analgesic or anti-inflammatory activity, respectively, and completely devoid of acute gastrolesivity. 155
Analogs, formulations and derivatives of imatinib: A patent review 143
Mechanisms involved in the antiplatelet activity of 8-methyl-4-(1-piperazinyl)-7-(3-pyridinylmethoxy)-2H-1-benzopyran-2-one (RC414) 139
Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma 133
1,5-Benzodiazepine tricyclic derivatives exerting anti-inflammatory effects in mice by inhibiting interleukin-6 and prostaglandin E2 production 132
1,5-Benzodiazepines. Part XIII. Substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines and 4H-imidazo[1,2-a][1,5]benzodiazepin-5-amines as analgesic, anti-inflammatory and/or antipyretic agents with low acute toxicity 131
Modulation of native GABAA receptor activity by triazolo 1,5-benzodiazepines 131
1,8-Naphthyridines IV. 9-substituted N,N-dialkyl-5-(alkylamino or cycloalkylamino) [1,2,4]triazolo[4,3-a][1, 8]naphthyridine-6-carboxamides, new compounds with anti-aggressive and potent anti-inflammatory activities 130
null 128
1,5-Benzodiazepines XIV. Synthesis of new substituted 9H-bis[1,2,4]triazolo[4,3-a:3',4'-d][1,5]benzodiazepines and related compounds endowed with in vitro cytotoxic properties 126
Coumarin, chromone, and 4(3H)-pyrimidinone novel bicyclic and tricyclic derivatives as antiplatelet agents: synthesis, biological evaluation and comparative molecular field analysis 126
1,8-Naphthyridines V.Novel N-substituted 5-amino-N,N-diethyl-9-isopropyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, as potent anti-inflammatory and/or analgesic agents completely devoid of acute gastrolesivity 124
Anticonvulsive Activity in Audiogenic DBA/2 Mice of 1,4-Benzodiazepines and 1,5-Benzodiazepines with Different Activities at Cerebellar Granule Cell GABAA Receptors 124
1,8-Naphthyridines VII. New substituted 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides and their isosteric analogues, exhibiting notable anti-inflammatory and/or analgesic activities, but no acute gastrolesivity 123
1,8-Naphthyridines VI. Synthesis and anti-inflammatory activity of 5-(alkylamino)-N,N-diethyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6 carboxamides with a new substitution pattern on the triazole ring 121
Solvent-free reactions as green chemistry procedures for the synthesis of cosmetic fatty esters 117
Study of the Interaction of 1,4- and 1,5-Benzodiazepines with GABAA Receptors of Rat Cerebellum Granule Cells in Culture 114
Conjugated Methyl Sulfide and Phenyl Sulfide Derivatives of Oxidosqualene as Inhibitors of Oxidosqualene and Squalene-Hopene Cyclases 114
Efficient one-pot synthesis of N-substituted 2-aminochromones, their benzo-fused derivatives, and diaminobenzodipyrandiones of two new structural classes 113
Synthesis of (E)- and (Z)-29-methylidyne-2,3-oxidosqualene derivatives as inhibitors of liver and yeast oxidosqualene cyclase 109
Recent Studies on Ponatinib in Cancers Other Than Chronic Myeloid Leukemia 107
Fine molecular tuning at position 4 of 2H-chromen-2-one derivatives in the search of potent and selective monoamine oxidase B inhibitors 103
New 1,5 - Benzodiazepine Compounds: Activity at Native GABAA Receptors 102
Synthesis, antiplatelet activity and comparative molecular fields analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues 101
Synthesis and in vitro antiplatelet activity of new 4-(1-piperazinyl)coumarin derivatives. Human platelet phosphodiesterase 3 inhibitory properties of the two most effective compounds described and molecular modeling study on their interactions with phosphodiesterase 3A catalytic site 101
Pyrrolo[2,3-d]pyrimidines as kinase inhibitors 101
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction 99
Pyran derivatives XX. 2-Aminochromone benzo-fused derivatives with antiproliferative properties 93
Mechanism of action of two new pyrimidoquinoline and isoquinoline derivatives in human platelets 90
1,5-Benzodiazepines. Part XII. Synthesis and biological evaluation of tricyclic and tetracyclic 1,5-benzodiazepines derivatives as nevirapine analogues 88
Pyran derivatives. Part XXI. Antiproliferative and cytotoxic properties of novel N-substituted 4-aminocoumarins, their benzo-fused derivatives, and some related 2-aminochromones 87
GABA A Receptors of Cerebellar Granule in Culture: Interaction with Benzodiazepines 86
1,5-Benzodiazepines. X. Dialkylamino substituted 1,5-benzodiazepine and [1,2,4]triazolo[4,3-a][1,5]benzodiazepine derivatives with inhibitory activity on PAF-induced platelet aggregation 84
An Update on JAK Inhibitors 84
3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors 81
Crystal structure of N,N-dimethyl-1-phenyl-4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amine, C18H17N5 72
1,8-Naphthyridines III. N,N-Dialkyl-5-chloro[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides with anti-inflammatory activity 69
Sinthesis in vitro inhibitory activity on human platelet aggregation of novel properly substituted 4-(1-piperazinyl)-coumarins 66
Acid-catalysed Hydrolisis and Benzodiazepine-like Properties of 5-(Dialkylamino)- and 5-(Alkylthio)-substituted 8-Chloro-6-phenyl-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepines in mice 66
Combining repositioning and de novo synthesis of pyrazolo[3,4-d]pyrimidines to discover potent SIRT-2 inhibitors 43
Insights into RNA-dependent RNA Polymerase Inhibitors as Anti-influenza Virus Agents 42
PYRAZOLO[3,4-d]PYRIMIDINE DERIVATIVES AS SIRTUIN INHIBITORS: DESIGN, SYNTHESIS AND PRELIMINARY in vitro EVALUATION 41
Anti-Survival Effect of SI306 and Its Derivatives on Human Glioblastoma Cells 37
Synthetic Heterocyclic Derivatives as Kinase Inhibitors Tested for the Treatment of Neuroblastoma 36
Small Molecule Tyrosine Kinase Inhibitors (TKIs) for Glioblastoma Treatment 34
Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling 34
Pyrazole[3,4-d]pyrimidine derivatives loaded into halloysite as potential CDK inhibitors 25
A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation 21
Erratum: Synthesis, antiplatelet activity and comparative molecular field analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues (Bioorganic and Medicinal Chemistry (2000) 8 (751) PII: S80968089600000109) 13
1,8-Naphthyridines IX. Potent anti-inflammatory and/or analgesic activity of a new group of substituted 5-amino[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides, of some their Mannich base derivatives and of one novel substituted 5-amino-10-oxo-10Hpyrimido[ 1,2-a][1,8]naphthyridine-6-carboxamide derivative 13
Progress of pharmaceutical technological and cosmetic research at Genoa university 11
Synthesis, antiplatelet activity and comparative molecular field analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues 7
Halloysite Nanotube-Based Delivery of Pyrazolo[3,4-d]pyrimidine Derivatives for Prostate and Bladder Cancer Treatment 3
Totale 5.188
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Categoria #
all - tutte 16.505
article - articoli 15.788
book - libri 0
conference - conferenze 717
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 33.010
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020820 0 0 0 0 0 0 193 85 117 206 163 56
2020/2021349 41 30 16 22 17 50 13 33 30 46 25 26
2021/2022679 28 48 47 88 33 32 37 152 43 71 23 77
2022/2023629 56 61 6 68 79 92 3 62 89 11 90 12
2023/2024371 15 35 11 53 25 24 17 16 32 25 39 79
2024/2025483 34 78 38 71 133 114 15 0 0 0 0 0
Totale 5.188