GROSSI, GIANCARLO
GROSSI, GIANCARLO
100006 - Dipartimento di Farmacia
1,2-Fused Pyrimidines. V. Synthesis of 1-Alkyl or Phenyl-2H-dipyrido-[1,2-a:2’, 3’-d]pyrimidine-2,5(1H)-diones
1992-01-01 Mario Di, Braccio; Giorgio, Roma; Grossi, Giancarlo; Giovanni, Ciarallo
1,5-Benzodiazepine tricyclic derivatives exerting anti-inflammatory effects in mice by inhibiting interleukin-6 and prostaglandin E2 production
2001-01-01 Fruscella, P.; Sottocorno, M.; DI BRACCIO, Mario; Diomede, L.; Piccardi, N.; Cagnotto, A.; Grossi, Giancarlo; Romano, M.; Mennini, T.; Roma, Giorgio
1,5-Benzodiazepines IX. A new route to substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines with analgesic and/or anti-inflammatory activities
1991-01-01 Roma, Giorgio; Grossi, Giancarlo; DI BRACCIO, Mario; Ghia, M.; Mattioli, Francesca
1,5-Benzodiazepines XIV. Synthesis of new substituted 9H-bis[1,2,4]triazolo[4,3-a:3',4'-d][1,5]benzodiazepines and related compounds endowed with in vitro cytotoxic properties
2005-01-01 DI BRACCIO, Mario; Grossi, Giancarlo; Ceruti, M.; Rocco, F.; Loddo, R.; Sanna, G.; Busonera, B.; Marreddu, M.; Marongiu, M. E.
1,5-Benzodiazepines. Part XII. Synthesis and biological evaluation of tricyclic and tetracyclic 1,5-benzodiazepines derivatives as nevirapine analogues
2001-01-01 Mario Di, Braccio; Grossi, Giancarlo; Giorgio, Roma; Laura, Vargiu; Massimo, Mura; Maria Elena, Marongiu
1,5-Benzodiazepines. Part XIII. Substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines and 4H-imidazo[1,2-a][1,5]benzodiazepin-5-amines as analgesic, anti-inflammatory and/or antipyretic agents with low acute toxicity
2002-01-01 Grossi, Giancarlo; DI BRACCIO, Mario; Roma, Giorgio; V., Ballabeni; M., Tognolini; F., Calcina; E., Barocelli
1,5-Benzodiazepines. X. Dialkylamino substituted 1,5-benzodiazepine and [1,2,4]triazolo[4,3-a][1,5]benzodiazepine derivatives with inhibitory activity on PAF-induced platelet aggregation
1992-01-01 Mario Di, Braccio; Giorgio, Roma; Grossi, Giancarlo; Giuliana, Leoncini; Mitzi, Maresca
1,8-Naphthyridines III. N,N-Dialkyl-5-chloro[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides with anti-inflammatory activity
1997-01-01 DI BRACCIO, Mario; Roma, Giorgio; Grossi, Giancarlo; Ghia, M.; Mattioli, Francesca
1,8-Naphthyridines IV. 9-substituted N,N-dialkyl-5-(alkylamino or cycloalkylamino) [1,2,4]triazolo[4,3-a][1, 8]naphthyridine-6-carboxamides, new compounds with anti-aggressive and potent anti-inflammatory activities
2000-01-01 Roma, Giorgio; DI BRACCIO, Mario; Grossi, Giancarlo; Mattioli, Francesca; Ghia, M.
1,8-Naphthyridines IX. Potent anti-inflammatory and/or analgesic activity of a new group of substituted 5-amino[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides, of some their Mannich base derivatives and of one novel substituted 5-amino-10-oxo-10Hpyrimido[ 1,2-a][1,8]naphthyridine-6-carboxamide derivative
2014-01-01 Mario Di Braccio, A; Grossi, Giancarlo; Alfei, Silvana; Vigilio Ballabeni, C; Massimiliano Tognolini, C; Lisa Flammini, C; Carmine Giorgio, C; Simona Bertoni, C; Elisabetta Barocelli, C.
1,8-Naphthyridines V.Novel N-substituted 5-amino-N,N-diethyl-9-isopropyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, as potent anti-inflammatory and/or analgesic agents completely devoid of acute gastrolesivity
2005-01-01 Grossi, Giancarlo; DI BRACCIO, Mario; Roma, Giorgio; Ballabeni, V.; Tognolini, M.; Barocelli, E.
1,8-Naphthyridines VI. Synthesis and anti-inflammatory activity of 5-(alkylamino)-N,N-diethyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6 carboxamides with a new substitution pattern on the triazole ring
2008-01-01 DI BRACCIO, Mario; Grossi, Giancarlo; Roma, Giorgio; D., Piras; Mattioli, Francesca; Gosmar, Marzia
1,8-Naphthyridines VII. New substituted 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides and their isosteric analogues, exhibiting notable anti-inflammatory and/or analgesic activities, but no acute gastrolesivity
2008-01-01 Roma, Giorgio; Grossi, Giancarlo; DI BRACCIO, Mario; Piras, D.; Ballabeni, V.; Tognolini, M.; Bertoni, S.; Barocelli, E.
1,8-Naphthyridines VIII. Novel 5-aminoimidazo[1,2-a][1,8]naphthyridine-6-carboxamide and 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamide derivatives showing potent analgesic or anti-inflammatory activity, respectively, and completely devoid of acute gastrolesivity.
2010-01-01 Giorgio, Roma; DI BRACCIO, Mario; Grossi, Giancarlo; Daniela, Piras; Vigilio, Ballabeni; Massimiliano, Tognolini; Simona, Bertoni; Elisabetta, Barocelli
3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors
2018-01-01 Giacchello, I.; Trist, I. M. L; Musumeci, F.; Greco, C.; D’Agostino, I.; Deodato, D.; Loregian, A.; Grossi, G.; Schenone, S.
A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation
2024-01-01 Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Brullo, C.; Musumeci, Francesca; Bruzzone, S.; Cichero, E.; Schenone, S.
Acid-catalysed Hydrolisis and Benzodiazepine-like Properties of 5-(Dialkylamino)- and 5-(Alkylthio)-substituted 8-Chloro-6-phenyl-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepines in mice
1998-01-01 Silvio, Caccia; Grossi, Giancarlo; Claudia, Fracasso; Angelo, Nacca; Alfredo, Cagnotto; Tiziana, Mennini; Marco, Ghia; Giorgio, Roma
An Update on JAK Inhibitors
2019-01-01 Musumeci, Francesca; Greco, Chiara; Giacchello, Ilaria; Fallacara, Anna Lucia; Ibrahim, Munjed M; Grossi, Giancarlo; Brullo, Chiara; Schenone, Silvia
Analogs, formulations and derivatives of imatinib: A patent review
2015-01-01 Musumeci, Francesca; Schenone, Silvia; Grossi, Giancarlo; Brullo, Chiara; Sanna, Monica
Anti-Survival Effect of SI306 and Its Derivatives on Human Glioblastoma Cells
2022-01-01 Monteleone, Lorenzo; Marengo, Barbara; Musumeci, Francesca; Grossi, Giancarlo; Carbone, Anna; Valenti, Giulia E.; Domenicotti, Cinzia; Schenone, Silvia