LUSARDI, MATTEO

LUSARDI, MATTEO  

100006 - Dipartimento di Farmacia  

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Titolo Data di pubblicazione Autore(i) File
Amino-Pyrazoles in Medicinal Chemistry: A Review 1-gen-2023 Lusardi, Matteo; Spallarossa, Andrea; Brullo, Chiara
AMINO-PYRAZOLES: A PRIVILEGED SCAFFOLD FOR THE SYNTHESIS OF BIOLOGICALLY ACTIVE COMPOUNDS 1-gen-2023 Lusardi, Matteo
Antimalarial Activity of Tri- and Tetra-Substituted Anilino Pyrazoles 1-gen-2023 Lusardi, Matteo; Basilico, Nicoletta; Rotolo, Chiara; Parapini, Silvia; Spallarossa, Andrea
Bicyclic basic merbarone analogues as antiproliferative agents 1-gen-2021 Spallarossa, A.; Lusardi, M.; Caneva, C.; Profumo, A.; Rosano, C.; Ponassi, M.
Cyclic diacyl thioureas enhance activity of corrector Lumacaftor on F508del‐CFTR 1-gen-2024 Spallarossa, Andrea; Pedemonte, Nicoletta; Pesce, Emanuela; Millo, Enrico; Cichero, Elena; Rosano, Camillo; Lusardi, Matteo; Iervasi, Erika; Ponassi, Marco
Design, synthesis and biological evaluation of novel 5-amino pyrazoles with antiangiogenic properties 1-gen-2022 Lusardi, Matteo; Brullo, Chiara; Ponassi, Marco; Wehrle-Haller, Bernhard; Spallarossa, Andrea
Diversity-oriented synthesis of highly-functionalized amino-pyrazoles as pharmaceutically relevant compounds 26-mar-2024 Lusardi, Matteo
HIGHLY-FUNCTIONALIZED AMINO PYRAZOLES AS ANTIOXIDANT AGENTS: A PRELIMINARY SYNTHETIC ACCESSIBILITY STUDY 1-gen-2021 Lusardi, Matteo; Brullo, Chiara; Spallarossa, Andrea
Novel 5-aminopyrazoles endowed with anti-angiogenetic properties: Design, synthesis and biological evaluation 1-gen-2023 Lusardi, Matteo; Wehrle-Haller, Bernhard; Sidibe, Adama; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea
Novel amino-pyrazole analogues interfering with cell migration 1-gen-2022 Lusardi, Matteo; Brullo, Chiara; Ponassi, Marco; Wehrle-Haller, Bernhard; Spallarossa, Andrea
One-Pot Synthesis and Antiproliferative Activity of Highly Functionalized Pyrazole Derivatives 1-gen-2022 Lusardi, M.; Rotolo, C.; Ponassi, M.; Iervasi, E.; Rosano, C.; Spallarossa, A.
Potent and Broad-Spectrum Bactericidal Activity of a Nanotechnologically Manipulated Novel Pyrazole 1-gen-2022 Alfei, Silvana; Caviglia, Debora; Zorzoli, Alessia; Marimpietri, Danilo; Spallarossa, Andrea; Lusardi, Matteo; Zuccari, Guendalina; Schito, Anna Maria
Regioselective synthesis and structural characterization of novel tri- and tetra- substituted anilino pyrazoles endowed with antimalarial activity 1-gen-2023 Lusardi, Matteo; Basilico, Nicoletta; Parapini, Silvia; Iervasi, Erika; Ponassi, Marco; Spallarossa, Andrea
Regioselective Synthesis, Structural Characterization, and Antiproliferative Activity of Novel Tetra-Substituted Phenylaminopyrazole Derivatives 1-gen-2022 Lusardi, Matteo; Profumo, Aldo; Rotolo, Chiara; Iervasi, Erika; Rosano, Camillo; Spallarossa, Andrea; Ponassi, Marco
Scouting in silico different chemo-types of PDE4 inhibitors to guide the design of new anti-inflammatory/antioxidant agents 1-gen-2023 Cichero, Elena; Rapetti, Federica; Lusardi, Matteo; Scarano, Naomi; Alfei, Silvana; Altieri, Paola; Garibaldi, Silvano; Ameri, Pietro; Signorello, MARIA GRAZIA; Brullo, Chiara
STRUCTURAL FUNCTIONALIZATION OF TRI-SUBSTITUTED PYRAZOLE DERIVATIVES AND PRELIMINARY EVALUATION OF THEIR ANTIMALARIAL ACTIVITY 1-gen-2023 Lusardi, M.; Basilico, N.; Parapini, S.; Iervasi, E; Ponassi, M.; Spallarossa, A
Successful Dendrimer and Liposome-Based Strategies to Solubilize an Antiproliferative Pyrazole Otherwise Not Clinically Applicable 1-gen-2022 Alfei, S.; Spallarossa, A.; Lusardi, M.; Zuccari, G.
Synthesis and biological evaluation of new pyrazole carbohydrazides as antiproliferative and antioxidant agents. 1-gen-2021 Lusardi, Matteo; Brullo, Chiara; Signorello, MARIA GRAZIA; Ponassi, Marco; Iervasi, Erika; Spallarossa, Andrea
Synthesis, Antiproliferative, and Antioxidant Properties of Highly Functionalized Pyrazoles 1-gen-2022 Lusardi, Matteo; Brullo, Chiara; Signorello, MARIA GRAZIA; Ponassi, Marco; Spallarossa, Andrea