LUSARDI, MATTEO
LUSARDI, MATTEO
100006 - Dipartimento di Farmacia
Amino-Pyrazoles in Medicinal Chemistry: A Review
2023-01-01 Lusardi, Matteo; Spallarossa, Andrea; Brullo, Chiara
AMINO-PYRAZOLES: A PRIVILEGED SCAFFOLD FOR THE SYNTHESIS OF BIOLOGICALLY ACTIVE COMPOUNDS
2023-01-01 Lusardi, Matteo
Antimalarial Activity of Tri- and Tetra-Substituted Anilino Pyrazoles
2023-01-01 Lusardi, Matteo; Basilico, Nicoletta; Rotolo, Chiara; Parapini, Silvia; Spallarossa, Andrea
Bicyclic basic merbarone analogues as antiproliferative agents
2021-01-01 Spallarossa, A.; Lusardi, M.; Caneva, C.; Profumo, A.; Rosano, C.; Ponassi, M.
Design, synthesis and biological evaluation of novel 5-amino pyrazoles with antiangiogenic properties
2022-01-01 Lusardi, Matteo; Brullo, Chiara; Ponassi, Marco; Wehrle-Haller, Bernhard; Spallarossa, Andrea
HIGHLY-FUNCTIONALIZED AMINO PYRAZOLES AS ANTIOXIDANT AGENTS: A PRELIMINARY SYNTHETIC ACCESSIBILITY STUDY
2021-01-01 Lusardi, Matteo; Brullo, Chiara; Spallarossa, Andrea
Novel 5-aminopyrazoles endowed with anti-angiogenetic properties: Design, synthesis and biological evaluation
2023-01-01 Lusardi, Matteo; Wehrle-Haller, Bernhard; Sidibe, Adama; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea
Novel amino-pyrazole analogues interfering with cell migration
2022-01-01 Lusardi, Matteo; Brullo, Chiara; Ponassi, Marco; Wehrle-Haller, Bernhard; Spallarossa, Andrea
One-Pot Synthesis and Antiproliferative Activity of Highly Functionalized Pyrazole Derivatives
2022-01-01 Lusardi, M.; Rotolo, C.; Ponassi, M.; Iervasi, E.; Rosano, C.; Spallarossa, A.
Potent and Broad-Spectrum Bactericidal Activity of a Nanotechnologically Manipulated Novel Pyrazole
2022-01-01 Alfei, Silvana; Caviglia, Debora; Zorzoli, Alessia; Marimpietri, Danilo; Spallarossa, Andrea; Lusardi, Matteo; Zuccari, Guendalina; Schito, Anna Maria
Regioselective synthesis and structural characterization of novel tri- and tetra- substituted anilino pyrazoles endowed with antimalarial activity
2023-01-01 Lusardi, Matteo; Basilico, Nicoletta; Parapini, Silvia; Iervasi, Erika; Ponassi, Marco; Spallarossa, Andrea
Regioselective Synthesis, Structural Characterization, and Antiproliferative Activity of Novel Tetra-Substituted Phenylaminopyrazole Derivatives
2022-01-01 Lusardi, Matteo; Profumo, Aldo; Rotolo, Chiara; Iervasi, Erika; Rosano, Camillo; Spallarossa, Andrea; Ponassi, Marco
Scouting in silico different chemo-types of PDE4 inhibitors to guide the design of new anti-inflammatory/antioxidant agents
2023-01-01 Cichero, Elena; Rapetti, Federica; Lusardi, Matteo; Scarano, Naomi; Alfei, Silvana; Altieri, Paola; Garibaldi, Silvano; Ameri, Pietro; Signorello, MARIA GRAZIA; Brullo, Chiara
STRUCTURAL FUNCTIONALIZATION OF TRI-SUBSTITUTED PYRAZOLE DERIVATIVES AND PRELIMINARY EVALUATION OF THEIR ANTIMALARIAL ACTIVITY
2023-01-01 Lusardi, M.; Basilico, N.; Parapini, S.; Iervasi, E; Ponassi, M.; Spallarossa, A
Successful Dendrimer and Liposome-Based Strategies to Solubilize an Antiproliferative Pyrazole Otherwise Not Clinically Applicable
2022-01-01 Alfei, S.; Spallarossa, A.; Lusardi, M.; Zuccari, G.
Synthesis and biological evaluation of new pyrazole carbohydrazides as antiproliferative and antioxidant agents.
2021-01-01 Lusardi, Matteo; Brullo, Chiara; Signorello, MARIA GRAZIA; Ponassi, Marco; Iervasi, Erika; Spallarossa, Andrea
Synthesis, Antiproliferative, and Antioxidant Properties of Highly Functionalized Pyrazoles
2022-01-01 Lusardi, Matteo; Brullo, Chiara; Signorello, MARIA GRAZIA; Ponassi, Marco; Spallarossa, Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Amino-Pyrazoles in Medicinal Chemistry: A Review | 1-gen-2023 | Lusardi, Matteo; Spallarossa, Andrea; Brullo, Chiara | |
AMINO-PYRAZOLES: A PRIVILEGED SCAFFOLD FOR THE SYNTHESIS OF BIOLOGICALLY ACTIVE COMPOUNDS | 1-gen-2023 | Lusardi, Matteo | |
Antimalarial Activity of Tri- and Tetra-Substituted Anilino Pyrazoles | 1-gen-2023 | Lusardi, Matteo; Basilico, Nicoletta; Rotolo, Chiara; Parapini, Silvia; Spallarossa, Andrea | |
Bicyclic basic merbarone analogues as antiproliferative agents | 1-gen-2021 | Spallarossa, A.; Lusardi, M.; Caneva, C.; Profumo, A.; Rosano, C.; Ponassi, M. | |
Design, synthesis and biological evaluation of novel 5-amino pyrazoles with antiangiogenic properties | 1-gen-2022 | Lusardi, Matteo; Brullo, Chiara; Ponassi, Marco; Wehrle-Haller, Bernhard; Spallarossa, Andrea | |
HIGHLY-FUNCTIONALIZED AMINO PYRAZOLES AS ANTIOXIDANT AGENTS: A PRELIMINARY SYNTHETIC ACCESSIBILITY STUDY | 1-gen-2021 | Lusardi, Matteo; Brullo, Chiara; Spallarossa, Andrea | |
Novel 5-aminopyrazoles endowed with anti-angiogenetic properties: Design, synthesis and biological evaluation | 1-gen-2023 | Lusardi, Matteo; Wehrle-Haller, Bernhard; Sidibe, Adama; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea | |
Novel amino-pyrazole analogues interfering with cell migration | 1-gen-2022 | Lusardi, Matteo; Brullo, Chiara; Ponassi, Marco; Wehrle-Haller, Bernhard; Spallarossa, Andrea | |
One-Pot Synthesis and Antiproliferative Activity of Highly Functionalized Pyrazole Derivatives | 1-gen-2022 | Lusardi, M.; Rotolo, C.; Ponassi, M.; Iervasi, E.; Rosano, C.; Spallarossa, A. | |
Potent and Broad-Spectrum Bactericidal Activity of a Nanotechnologically Manipulated Novel Pyrazole | 1-gen-2022 | Alfei, Silvana; Caviglia, Debora; Zorzoli, Alessia; Marimpietri, Danilo; Spallarossa, Andrea; Lusardi, Matteo; Zuccari, Guendalina; Schito, Anna Maria | |
Regioselective synthesis and structural characterization of novel tri- and tetra- substituted anilino pyrazoles endowed with antimalarial activity | 1-gen-2023 | Lusardi, Matteo; Basilico, Nicoletta; Parapini, Silvia; Iervasi, Erika; Ponassi, Marco; Spallarossa, Andrea | |
Regioselective Synthesis, Structural Characterization, and Antiproliferative Activity of Novel Tetra-Substituted Phenylaminopyrazole Derivatives | 1-gen-2022 | Lusardi, Matteo; Profumo, Aldo; Rotolo, Chiara; Iervasi, Erika; Rosano, Camillo; Spallarossa, Andrea; Ponassi, Marco | |
Scouting in silico different chemo-types of PDE4 inhibitors to guide the design of new anti-inflammatory/antioxidant agents | 1-gen-2023 | Cichero, Elena; Rapetti, Federica; Lusardi, Matteo; Scarano, Naomi; Alfei, Silvana; Altieri, Paola; Garibaldi, Silvano; Ameri, Pietro; Signorello, MARIA GRAZIA; Brullo, Chiara | |
STRUCTURAL FUNCTIONALIZATION OF TRI-SUBSTITUTED PYRAZOLE DERIVATIVES AND PRELIMINARY EVALUATION OF THEIR ANTIMALARIAL ACTIVITY | 1-gen-2023 | Lusardi, M.; Basilico, N.; Parapini, S.; Iervasi, E; Ponassi, M.; Spallarossa, A | |
Successful Dendrimer and Liposome-Based Strategies to Solubilize an Antiproliferative Pyrazole Otherwise Not Clinically Applicable | 1-gen-2022 | Alfei, S.; Spallarossa, A.; Lusardi, M.; Zuccari, G. | |
Synthesis and biological evaluation of new pyrazole carbohydrazides as antiproliferative and antioxidant agents. | 1-gen-2021 | Lusardi, Matteo; Brullo, Chiara; Signorello, MARIA GRAZIA; Ponassi, Marco; Iervasi, Erika; Spallarossa, Andrea | |
Synthesis, Antiproliferative, and Antioxidant Properties of Highly Functionalized Pyrazoles | 1-gen-2022 | Lusardi, Matteo; Brullo, Chiara; Signorello, MARIA GRAZIA; Ponassi, Marco; Spallarossa, Andrea |