Sfoglia per Autore
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents
2014-01-01 Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines
2014-01-01 Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Anna, Sparatore; Boido, Vito; Sparatore, Fabio; Sara, Cannas; Paola, Molicotti; Stefania, Zanetti; Silvia, Parapini; Roberta, Loddo
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5
2015-01-01 Roberta, Loddo; Novelli, Federica; Anna, Sparatore; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Gabriella, Collu; Ilenia, Delogu; Gabriele, Giliberti; Paolo, La Colla
Synthesis and antiplasmodial activity of novel chloroquine analogues with bulky basic side chains
2015-01-01 Tasso, Bruno; Novelli, Federica; Tonelli, Michele; Barteselli, Anna; Basilico, Nicoletta; Parapini, Silvia; Taramelli, Donatella; Sparatore, Anna; Sparatore, Fabio
Multitarget Therapeutic Leads for Alzheimer’s Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and beta-Amyloid (Abeta) Aggregation
2015-01-01 Tonelli, Michele; Catto, Marco*; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Iusco, Giovanna; Pisani, Leonardo; De Stradis, Angelo; Denora, Nunzio; Sparatore, Anna; Boido, Vito; Carotti, Angelo; Sparatore, Fabio
Clofazimine analogs with antileishmanial and antiplasmodial activity
2015-01-01 Barteselli, A.; Casagrande, M.; Basilico, N.; Parapini, S.; Rusconi, C. M.; Tonelli, Michele; Boido, Vito; Taramelli, D.; Sparatore, Fabio; Sparatore, A.
Fight against H1N1 Influenza A Virus: Recent Insights towards the Development of Druggable Compounds
2016-01-01 Tonelli, Michele; Cichero, Elena
Celecoxib Inhibits Prion Protein 90-231-Mediated Pro-inflammatory Responses in Microglial Cells
2016-01-01 Villa, Valentina; THELLUNG DE COURTELARY, Stefano; Corsaro, Alessandro; Novelli, Federica; Tasso, Bruno; Colucci D’Amato, L.; Gatta, Elena; Tonelli, Michele; Florio, Tullio
Novel celecoxib analogues inhibit glial production of prostaglandinE2, nitric oxide, and oxygen radicals reverting the neuroinflammatoryresponses induced by misfolded prion protein fragment 90-231 or lipopolysaccharide
2016-01-01 Villa, Valentina; THELLUNG DE COURTELARY, Stefano; Bajetto, Adriana; Gatta, Elena; Robello, Mauro; Novelli, Federica; Tasso, Bruno; Tonelli, Michele; Florio, Tullio
Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles
2017-01-01 Cichero, Elena; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Delogu, I; Loddo, R.; Bruno, Olga; Fossa, Paola
Host DHFR-directed cycloguanil analogues endowed with promising activity against influenza virus and respiratory syncytial virus
2017-01-01 Tonelli, Michele
Novel biguanide-based derivatives scouted as TAAR1 agonists: synthesis, biological evaluation, ADME prediction and molecular docking studies
2017-01-01 Tonelli, Michele; Espinoza, Stefano; Gainetdinov, RauL R.; Cichero, Elena
Targeting species-specific TAAR1 ligands: to date perspective of the rational drug design process
2017-01-01 Cichero, Elena; Tonelli, Michele
New insights into the structure of the Trace Amine-Associated Receptor 2 (TAAR2): homology modeling studies exploring the binding mode of 3-iodothyronamine
2017-01-01 Cichero, Elena; Tonelli, Michele
New arylsparteine derivatives as positive inotropic drugs
2017-01-01 Boido, Vito; Ercoli, Marcella; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Sparatore, Fabio; Cichero, Elena; Fossa, Paola; Dorigo, Paola; Froldi, Guglielmina
Host dihydrofolate reductase (DHFR)-directed cycloguanil analogues endowed with activity against influenza virus and respiratory syncytial virus
2017-01-01 Tonelli, Michele; Naesens, Lieve; Gazzarrini, Sabrina; Santucci, Matteo; Cichero, Elena; Tasso, Bruno; Moroni, Anna; Costi, Maria Paola; Loddo, Roberta
Exhaustive CoMFA and CoMSIA analyses around different chemical entities: a ligand-based study exploring the affinity and selectivity profiles of 5-HT1A ligands
2017-01-01 Guariento, S. .; Franchini, S.; Tonelli, Michele; Fossa, Paola; Sorbi, C.; Cichero, Elena; Brasili, L.
Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR)
2018-01-01 Francesconi, Valeria; Luca, Giovannini; Santucci, Matteo; Cichero, Elena; Paola Costi, Maria; Naesens, Lieve; Giordanetto, Fabrizio; Tonelli, Michele
9-Aminoacridine-based agents impair the bovine viral diarrhea virus (BVDV) replication targeting the RNA-dependent RNA polymerase (RdRp)
2018-01-01 Loddo, Roberta; Francesconi, Valeria; Laurini, Erik; Boccardo, Silvia; Aulic, Suzana; Fermeglia, Maurizio; Pricl, Sabrina; Tonelli, Michele
Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction
2018-01-01 Tonelli, Michele; Cichero, Elena; Mokhtar Mahmoud, Alì; Rabbito, Alessandro; Tasso, Bruno; Fossa, Paola; Ligresti, Alessia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents | 1-gen-2014 | Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta | |
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines | 1-gen-2014 | Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Anna, Sparatore; Boido, Vito; Sparatore, Fabio; Sara, Cannas; Paola, Molicotti; Stefania, Zanetti; Silvia, Parapini; Roberta, Loddo | |
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5 | 1-gen-2015 | Roberta, Loddo; Novelli, Federica; Anna, Sparatore; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Gabriella, Collu; Ilenia, Delogu; Gabriele, Giliberti; Paolo, La Colla | |
Synthesis and antiplasmodial activity of novel chloroquine analogues with bulky basic side chains | 1-gen-2015 | Tasso, Bruno; Novelli, Federica; Tonelli, Michele; Barteselli, Anna; Basilico, Nicoletta; Parapini, Silvia; Taramelli, Donatella; Sparatore, Anna; Sparatore, Fabio | |
Multitarget Therapeutic Leads for Alzheimer’s Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and beta-Amyloid (Abeta) Aggregation | 1-gen-2015 | Tonelli, Michele; Catto, Marco*; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Iusco, Giovanna; Pisani, Leonardo; De Stradis, Angelo; Denora, Nunzio; Sparatore, Anna; Boido, Vito; Carotti, Angelo; Sparatore, Fabio | |
Clofazimine analogs with antileishmanial and antiplasmodial activity | 1-gen-2015 | Barteselli, A.; Casagrande, M.; Basilico, N.; Parapini, S.; Rusconi, C. M.; Tonelli, Michele; Boido, Vito; Taramelli, D.; Sparatore, Fabio; Sparatore, A. | |
Fight against H1N1 Influenza A Virus: Recent Insights towards the Development of Druggable Compounds | 1-gen-2016 | Tonelli, Michele; Cichero, Elena | |
Celecoxib Inhibits Prion Protein 90-231-Mediated Pro-inflammatory Responses in Microglial Cells | 1-gen-2016 | Villa, Valentina; THELLUNG DE COURTELARY, Stefano; Corsaro, Alessandro; Novelli, Federica; Tasso, Bruno; Colucci D’Amato, L.; Gatta, Elena; Tonelli, Michele; Florio, Tullio | |
Novel celecoxib analogues inhibit glial production of prostaglandinE2, nitric oxide, and oxygen radicals reverting the neuroinflammatoryresponses induced by misfolded prion protein fragment 90-231 or lipopolysaccharide | 1-gen-2016 | Villa, Valentina; THELLUNG DE COURTELARY, Stefano; Bajetto, Adriana; Gatta, Elena; Robello, Mauro; Novelli, Federica; Tasso, Bruno; Tonelli, Michele; Florio, Tullio | |
Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles | 1-gen-2017 | Cichero, Elena; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Delogu, I; Loddo, R.; Bruno, Olga; Fossa, Paola | |
Host DHFR-directed cycloguanil analogues endowed with promising activity against influenza virus and respiratory syncytial virus | 1-gen-2017 | Tonelli, Michele | |
Novel biguanide-based derivatives scouted as TAAR1 agonists: synthesis, biological evaluation, ADME prediction and molecular docking studies | 1-gen-2017 | Tonelli, Michele; Espinoza, Stefano; Gainetdinov, RauL R.; Cichero, Elena | |
Targeting species-specific TAAR1 ligands: to date perspective of the rational drug design process | 1-gen-2017 | Cichero, Elena; Tonelli, Michele | |
New insights into the structure of the Trace Amine-Associated Receptor 2 (TAAR2): homology modeling studies exploring the binding mode of 3-iodothyronamine | 1-gen-2017 | Cichero, Elena; Tonelli, Michele | |
New arylsparteine derivatives as positive inotropic drugs | 1-gen-2017 | Boido, Vito; Ercoli, Marcella; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Sparatore, Fabio; Cichero, Elena; Fossa, Paola; Dorigo, Paola; Froldi, Guglielmina | |
Host dihydrofolate reductase (DHFR)-directed cycloguanil analogues endowed with activity against influenza virus and respiratory syncytial virus | 1-gen-2017 | Tonelli, Michele; Naesens, Lieve; Gazzarrini, Sabrina; Santucci, Matteo; Cichero, Elena; Tasso, Bruno; Moroni, Anna; Costi, Maria Paola; Loddo, Roberta | |
Exhaustive CoMFA and CoMSIA analyses around different chemical entities: a ligand-based study exploring the affinity and selectivity profiles of 5-HT1A ligands | 1-gen-2017 | Guariento, S. .; Franchini, S.; Tonelli, Michele; Fossa, Paola; Sorbi, C.; Cichero, Elena; Brasili, L. | |
Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR) | 1-gen-2018 | Francesconi, Valeria; Luca, Giovannini; Santucci, Matteo; Cichero, Elena; Paola Costi, Maria; Naesens, Lieve; Giordanetto, Fabrizio; Tonelli, Michele | |
9-Aminoacridine-based agents impair the bovine viral diarrhea virus (BVDV) replication targeting the RNA-dependent RNA polymerase (RdRp) | 1-gen-2018 | Loddo, Roberta; Francesconi, Valeria; Laurini, Erik; Boccardo, Silvia; Aulic, Suzana; Fermeglia, Maurizio; Pricl, Sabrina; Tonelli, Michele | |
Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction | 1-gen-2018 | Tonelli, Michele; Cichero, Elena; Mokhtar Mahmoud, Alì; Rabbito, Alessandro; Tasso, Bruno; Fossa, Paola; Ligresti, Alessia |
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