Sfoglia per Autore
Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR)
2018-01-01 Francesconi, Valeria; Luca, Giovannini; Santucci, Matteo; Cichero, Elena; Paola Costi, Maria; Naesens, Lieve; Giordanetto, Fabrizio; Tonelli, Michele
Benzimidazole derivatives endowed with potent antileishmanial activity
2018-01-01 Tonelli, Michele; Gabriele, Elena; Piazza, Francesca; Basilico, Nicoletta; Parapini, Silvia; Tasso, Bruno; Loddo, Roberta; Sparatore, Fabio; Sparatore, Anna
Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction
2018-01-01 Tonelli, Michele; Cichero, Elena; Mokhtar Mahmoud, Alì; Rabbito, Alessandro; Tasso, Bruno; Fossa, Paola; Ligresti, Alessia
Quinone-based derivatives: a new class of multi-target agents against Alzheimer’s disease
2019-01-01 Campora, Marta; Catto, Marco; Relini, Annalisa; Canale, Claudio; Tasso, Bruno; Tonelli, Michele
New naphtho- and anthraquinone derivatives as Cholinesterase inhibitors for the treatment of Alzheimer's disease
2019-01-01 Campora, Marta; Marco, Catto; Tonelli, Michele; Tasso, Bruno
Pyrazole and imidazo[1,2-b]pyrazole derivatives as new potential anti-tuberculosis agents.
2019-01-01 Meta, E; Brullo, C; Tonelli, M; Franzblau, Sg; Wang, Y; Ma, R; Baojie, W; Orena, Bs; Pasca, MARIA ROSALIA; Bruno, O.
Trace amine associated receptor 1 (TAAR1) modulators: a patent review (2010-present)
2020-01-01 Tonelli, Michele; Cichero, Elena
Exploring the selectivity profile of sigma receptor ligands by molecular docking and pharmacophore analyses.
2020-01-01 Righetti, G.; Tonelli, M.; Fossa, P.; Cichero, E.
Novel 1-amidino-4-phenylpiperazines as potent agonists at human taar1 receptor: Rational design, synthesis, biological evaluation and molecular docking studies
2020-01-01 Francesconi, V.; Cichero, E.; Kanov, E. V.; Laurini, E.; Pricl, S.; Gainetdinov, R. R.; Tonelli, M.
Synthesis and biological evaluation of novel (thio)semicarbazone-based benzimidazoles as antiviral agents against human respiratory viruses
2020-01-01 Francesconi, Valeria; Cichero, Elena; Schenone, Silvia; Naesens, Lieve; Tonelli, Michele
New insights into the binding features of f508del cftr potentiators: A molecular docking, pharmacophore mapping and qsar analysis approach
2020-01-01 Righetti, G.; Casale, M.; Tonelli, M.; Liessi, N.; Fossa, P.; Pedemonte, N.; Millo, E.; Cichero, E.
Molecular Docking and QSAR Studies as Computational Tools Exploring the Rescue Ability of F508del CFTR Correctors
2020-01-01 Righetti, G.; Casale, M.; Liessi, N.; Tasso, B.; Salis, A.; Tonelli, M.; Millo, E.; Pedemonte, N.; Fossa, P.; Cichero, E.
Quinolizidine-derived lucanthone and amitriptyline analogues endowed with potent antileishmanial activity
2020-01-01 Tonelli, M.; Sparatore, A.; Basilico, N.; Cavicchini, L.; Parapini, S.; Tasso, B.; Laurini, E.; Pricl, S.; Boido, V.; Sparatore, F.
Probing In Silico the Benzimidazole Privileged Scaffold for the Development of Drug-like Anti-RSV Agents
2021-01-01 Cichero, Elena; Calautti, Alessio; Francesconi, Valeria; Tonelli, Michele; Schenone, Silvia; Fossa, Paola
Journey on naphthoquinone and anthraquinone derivatives: New insights in alzheimer’s disease
2021-01-01 Campora, M.; Francesconi, V.; Schenone, S.; Tasso, B.; Tonelli, M.
Multitarget Biological Profiling of New Naphthoquinone and Anthraquinone-Based Derivatives for the Treatment of Alzheimer's Disease
2021-01-01 Campora, M.; Canale, C.; Gatta, E.; Tasso, B.; Laurini, E.; Relini, A.; Pricl, S.; Catto, M.; Tonelli, M.
Optimization of the clofazimine structure leads to a highly water-soluble C3-aminopyridinyl riminophenazine endowed with improved anti-Wnt and anti-cancer activity in vitro and in vivo
2021-01-01 Koval, A.; Bassanini, I.; Xu, J.; Tonelli, M.; Boido, V.; Sparatore, F.; Amant, F.; Annibali, D.; Leucci, E.; Sparatore, A.; Katanaev, V. L.
Evidence of pyrimethamine and cycloguanil analogues as dual inhibitors of trypanosoma brucei pteridine reductase and dihydrofolate reductase
2021-01-01 Tassone, G.; Landi, G.; Linciano, P.; Francesconi, V.; Tonelli, M.; Tagliazucchi, L.; Costi, M. P.; Mangani, S.; Pozzi, C.
Magnolol and Luteolin Inhibition of α-Glucosidase Activity: Kinetics and Type of Interaction Detected by In Vitro and In Silico Studies
2022-01-01 Djeujo, F. M.; Ragazzi, E.; Urettini, M.; Sauro, B.; Cichero, E.; Tonelli, M.; Froldi, G.
Anti-α-glucosidase and antiglycation activities of α-mangostin and new xanthenone derivatives: Enzymatic kinetics and mechanistic insights through in vitro studies
2022-01-01 Djeujo, F. M.; Francesconi, V.; Gonella, M.; Ragazzi, E.; Tonelli, M.; Froldi, G.
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