Sfoglia per Autore
SGK1 as a new target for anticancer agents: a hit-to-lead study
2017-01-01 Musumeci, F.; Greco, C.; Alcaro, S.; Ortuso, F.; Perrotti, N.; Schenone, S.
Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists.
2017-01-01 Giacchello, I.; Musumeci, F.; Greco, C.; Sanna, M.; Schenone, S.; Trincavelli, M. L.; Tuccinardi, T.
Pyrrolo[2,3-d]pyrimidines as kinase inhibitors
2017-01-01 Musumeci, Francesca; Sanna, Monica; Grossi, Giancarlo; Brullo, Chiara; Fallacara, Anna Lucia; Schenone, Silvia
Matrine in association with FD‑2 stimulates F508del‑cystic fibrosis transmembrane conductance regulator activity in the presence of corrector VX809
2017-01-01 Marengo, Barbara; Speciale, Andrea; Senatore, Lisa; Garibaldi, Silvano; Musumeci, Francesca; Nieddu, Erika; Pollarolo, Benedetta; Pronzato, MARIA ADELAIDE; Schenone, Silvia; Mazzei, Mauro; Domenicotti, CINZIA MARIA
Pyrrolo[2,3-d]pyrimidines active as Btk inhibitors
2017-01-01 Musumeci, Francesca; Sanna, Monica; Greco, Chiara; Giacchello, Ilaria; Fallacara, Anna Lucia; Amato, Rosario; Schenone, Silvia
Prodrugs of Pyrazolo[3,4-d]pyrimidines: From Library Synthesis to Evaluation as Potential Anticancer Agents in an Orthotopic Glioblastoma Model
2017-01-01 Vignaroli, Giulia; Iovenitti, Giulia; Zamperini, Claudio; Coniglio, Federica; Calandro, Pierpaolo; Molinari, Alessio; Fallacara, Anna Lucia; Sartucci, Andrea; Calgani, Alessia; Colecchia, David; Mancini, Andrea; Festuccia, Claudio; Dreassi, Elena; Valoti, Massimo; Musumeci, Francesca; Chiariello, Mario; Angelucci, Adriano; Botta, Maurizio; Schenone, Silvia
Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma
2017-01-01 Musumeci, F; Fallacara, Al; Brullo, C; Grossi, G; Botta, L; Calandro, P; Chiariello, M; Kissova, M; Crespan, E; Maga, G; Schenone, S.
Synthesis of a small library of potential SGK1 inihibitors
2018-01-01 Greco, C.; Musumeci, F.; Giacchello, I.; Perrotti, N.; Alcaro, S.; Ortuso, F.; Schenone, S.
Pyrazolo[3,4-d]pyrimidines as tyrosine kinase inhibitors: synthesis and biological evaluation
2018-01-01 Musumeci, F.; Greco, C.; Giacchello, I.; Crespan, E.; Maga, G.; Schenone, S.; Fallacara, A. L.; Molinari, A.; Botta, M.
Pyrazolo[3,4-d]pyrimidine active on neuroblastoma cells
2018-01-01 Greco, C.; Musumeci, F.; Giacchello, I.; Gorjòn de Pablo, G.; Molinari, A.; Fallacara, A. L.; Di Maria, S.; Marengo, B.; Domenicotti, C.; Botta, M.; Schenone, S.
3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors
2018-01-01 Giacchello, I.; Trist, I. M. L; Musumeci, F.; Greco, C.; D’Agostino, I.; Deodato, D.; Loregian, A.; Grossi, G.; Schenone, S.
Exploring SAR of a new generation of pyrazolo[3,4-d]pyrimidines as Fyn tyrosine kinase inhibitors
2018-01-01 Musumeci, F.; Greco, Chiara; Navarro Pinin, L.; Giacchello, Ilaria; Crespan, E.; Passannanti, R.; Trist, I. M. L.; Maga, G.; Schenone, S.; Botta, M.
Water Solubility Enhancement of Pyrazolo[3,4-d]pyrimidine Derivatives via Miniaturized Polymer–Drug Microarrays
2018-01-01 Sanna, Monica; Sicilia, Giovanna; Alazzo, Ali; Singh, Nishant; Musumeci, Francesca; Schenone, Silvia; Spriggs, Keith A.; Burley, Jonathan C.; Garnett, Martin C.; Taresco, Vincenzo; Alexander, Cameron
Optimization of Aminoimidazole Derivatives as Src Family Kinase Inhibitors
2018-01-01 Francini, Cinzia Maria; Musumeci, Francesca; Fallacara, Anna Lucia; Botta, Lorenzo; Molinari, Alessio; Artusi, Roberto; Mennuni, Laura; Angelucci, Adriano; Schenone, Silvia
Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatment
2018-01-01 Molinari, Alessio; Fallacara, Anna Lucia; Di Maria, Salvatore; Zamperini, Claudio; Poggialini, Federica; Musumeci, Francesca; Schenone, Silvia; Angelucci, Adriano; Colapietro, Alessandro; Crespan, Emmanuele; Kissova, Miroslava; Maga, Giovanni; Botta, Maurizio
Recent Studies on Ponatinib in Cancers Other Than Chronic Myeloid Leukemia
2018-01-01 Musumeci, F; Greco, C; Grossi, G; Molinari, A; Schenone, S
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction
2018-01-01 D'Agostino, Ilaria; Giacchello, Ilaria; Nannetti, Giulio; Fallacara, Anna Lucia; Deodato, Davide; Musumeci, Francesca; Grossi, Giancarlo; Palù, Giorgio; Cau, Ylenia; Trist, Iuni Margaret; Loregian, Arianna; Schenone, Silvia; Botta, Maurizio
Formulation Of Pyrazolo[3,4-d]pyrimidines Kinase Inhibitors For The Treatment Of Glioblastoma Multiforme
2019-01-01 Greco, Chiara; Cavanagh, Robert; Taresco, Vincenzo; Vasey, Catherine; Musumeci, Francesca; Rahman, Ruman; Alexander, Cameron; Schenone, Silvia
The small molecule SI113 hinders epithelial-to-mesenchymal transition and subverts cytoskeletal organization in human cancer cells
2019-01-01 Abbruzzese, C.; Matteoni, S.; Persico, M.; Ascione, B.; Schenone, S.; Musumeci, F.; Amato, R.; Perrotti, N.; Matarrese, P.; Paggi, M. G.
Identification of a new family of pyrazolo[3,4-d]pyrimidine derivatives as multitarget Fyn-Blk-Lyn inhibitors active on B- and T-lymphoma cell lines
2019-01-01 Fallacara, A. L.; Passannanti, R.; Mori, M.; Iovenitti, G.; Musumeci, F.; Greco, C.; Crespan, E.; Kissova, M.; Maga, G.; Tarantelli, C.; Spriano, F.; Gaudio, E.; Bertoni, F.; Botta, M.; Schenone, S.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
SGK1 as a new target for anticancer agents: a hit-to-lead study | 1-gen-2017 | Musumeci, F.; Greco, C.; Alcaro, S.; Ortuso, F.; Perrotti, N.; Schenone, S. | |
Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists. | 1-gen-2017 | Giacchello, I.; Musumeci, F.; Greco, C.; Sanna, M.; Schenone, S.; Trincavelli, M. L.; Tuccinardi, T. | |
Pyrrolo[2,3-d]pyrimidines as kinase inhibitors | 1-gen-2017 | Musumeci, Francesca; Sanna, Monica; Grossi, Giancarlo; Brullo, Chiara; Fallacara, Anna Lucia; Schenone, Silvia | |
Matrine in association with FD‑2 stimulates F508del‑cystic fibrosis transmembrane conductance regulator activity in the presence of corrector VX809 | 1-gen-2017 | Marengo, Barbara; Speciale, Andrea; Senatore, Lisa; Garibaldi, Silvano; Musumeci, Francesca; Nieddu, Erika; Pollarolo, Benedetta; Pronzato, MARIA ADELAIDE; Schenone, Silvia; Mazzei, Mauro; Domenicotti, CINZIA MARIA | |
Pyrrolo[2,3-d]pyrimidines active as Btk inhibitors | 1-gen-2017 | Musumeci, Francesca; Sanna, Monica; Greco, Chiara; Giacchello, Ilaria; Fallacara, Anna Lucia; Amato, Rosario; Schenone, Silvia | |
Prodrugs of Pyrazolo[3,4-d]pyrimidines: From Library Synthesis to Evaluation as Potential Anticancer Agents in an Orthotopic Glioblastoma Model | 1-gen-2017 | Vignaroli, Giulia; Iovenitti, Giulia; Zamperini, Claudio; Coniglio, Federica; Calandro, Pierpaolo; Molinari, Alessio; Fallacara, Anna Lucia; Sartucci, Andrea; Calgani, Alessia; Colecchia, David; Mancini, Andrea; Festuccia, Claudio; Dreassi, Elena; Valoti, Massimo; Musumeci, Francesca; Chiariello, Mario; Angelucci, Adriano; Botta, Maurizio; Schenone, Silvia | |
Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma | 1-gen-2017 | Musumeci, F; Fallacara, Al; Brullo, C; Grossi, G; Botta, L; Calandro, P; Chiariello, M; Kissova, M; Crespan, E; Maga, G; Schenone, S. | |
Synthesis of a small library of potential SGK1 inihibitors | 1-gen-2018 | Greco, C.; Musumeci, F.; Giacchello, I.; Perrotti, N.; Alcaro, S.; Ortuso, F.; Schenone, S. | |
Pyrazolo[3,4-d]pyrimidines as tyrosine kinase inhibitors: synthesis and biological evaluation | 1-gen-2018 | Musumeci, F.; Greco, C.; Giacchello, I.; Crespan, E.; Maga, G.; Schenone, S.; Fallacara, A. L.; Molinari, A.; Botta, M. | |
Pyrazolo[3,4-d]pyrimidine active on neuroblastoma cells | 1-gen-2018 | Greco, C.; Musumeci, F.; Giacchello, I.; Gorjòn de Pablo, G.; Molinari, A.; Fallacara, A. L.; Di Maria, S.; Marengo, B.; Domenicotti, C.; Botta, M.; Schenone, S. | |
3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors | 1-gen-2018 | Giacchello, I.; Trist, I. M. L; Musumeci, F.; Greco, C.; D’Agostino, I.; Deodato, D.; Loregian, A.; Grossi, G.; Schenone, S. | |
Exploring SAR of a new generation of pyrazolo[3,4-d]pyrimidines as Fyn tyrosine kinase inhibitors | 1-gen-2018 | Musumeci, F.; Greco, Chiara; Navarro Pinin, L.; Giacchello, Ilaria; Crespan, E.; Passannanti, R.; Trist, I. M. L.; Maga, G.; Schenone, S.; Botta, M. | |
Water Solubility Enhancement of Pyrazolo[3,4-d]pyrimidine Derivatives via Miniaturized Polymer–Drug Microarrays | 1-gen-2018 | Sanna, Monica; Sicilia, Giovanna; Alazzo, Ali; Singh, Nishant; Musumeci, Francesca; Schenone, Silvia; Spriggs, Keith A.; Burley, Jonathan C.; Garnett, Martin C.; Taresco, Vincenzo; Alexander, Cameron | |
Optimization of Aminoimidazole Derivatives as Src Family Kinase Inhibitors | 1-gen-2018 | Francini, Cinzia Maria; Musumeci, Francesca; Fallacara, Anna Lucia; Botta, Lorenzo; Molinari, Alessio; Artusi, Roberto; Mennuni, Laura; Angelucci, Adriano; Schenone, Silvia | |
Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatment | 1-gen-2018 | Molinari, Alessio; Fallacara, Anna Lucia; Di Maria, Salvatore; Zamperini, Claudio; Poggialini, Federica; Musumeci, Francesca; Schenone, Silvia; Angelucci, Adriano; Colapietro, Alessandro; Crespan, Emmanuele; Kissova, Miroslava; Maga, Giovanni; Botta, Maurizio | |
Recent Studies on Ponatinib in Cancers Other Than Chronic Myeloid Leukemia | 1-gen-2018 | Musumeci, F; Greco, C; Grossi, G; Molinari, A; Schenone, S | |
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction | 1-gen-2018 | D'Agostino, Ilaria; Giacchello, Ilaria; Nannetti, Giulio; Fallacara, Anna Lucia; Deodato, Davide; Musumeci, Francesca; Grossi, Giancarlo; Palù, Giorgio; Cau, Ylenia; Trist, Iuni Margaret; Loregian, Arianna; Schenone, Silvia; Botta, Maurizio | |
Formulation Of Pyrazolo[3,4-d]pyrimidines Kinase Inhibitors For The Treatment Of Glioblastoma Multiforme | 1-gen-2019 | Greco, Chiara; Cavanagh, Robert; Taresco, Vincenzo; Vasey, Catherine; Musumeci, Francesca; Rahman, Ruman; Alexander, Cameron; Schenone, Silvia | |
The small molecule SI113 hinders epithelial-to-mesenchymal transition and subverts cytoskeletal organization in human cancer cells | 1-gen-2019 | Abbruzzese, C.; Matteoni, S.; Persico, M.; Ascione, B.; Schenone, S.; Musumeci, F.; Amato, R.; Perrotti, N.; Matarrese, P.; Paggi, M. G. | |
Identification of a new family of pyrazolo[3,4-d]pyrimidine derivatives as multitarget Fyn-Blk-Lyn inhibitors active on B- and T-lymphoma cell lines | 1-gen-2019 | Fallacara, A. L.; Passannanti, R.; Mori, M.; Iovenitti, G.; Musumeci, F.; Greco, C.; Crespan, E.; Kissova, M.; Maga, G.; Tarantelli, C.; Spriano, F.; Gaudio, E.; Bertoni, F.; Botta, M.; Schenone, S. |
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