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Preparation of ureidopyrazolecarboxylates with neutrophil chemotaxis inhibiting activity. 1-gen-2008 Bruno, Olga; Bondavalli, Francesco; Brullo, Chiara; Schenone, Silvia
Current advances in the development of anticancer drugs targeting tyrosine kinases of the Src family 1-gen-2008 Schenone, Silvia; Zanoli, S.; Brullo, Chiara; Crespan, E.; Maga, G.
Small molecules ATP-competitive inhibitors of FLT3: a chemical overview. 1-gen-2008 Schenone, Silvia; Brullo, Chiara; M., Botta
New pyrazolo[3,4-b]pyridines antagonist of A1 adenosine receptors 1-gen-2008 Schenone, Silvia; Brullo, Chiara; Bruno, Olga; Bondavalli, Francesco; Mosti, Luisa; Tuccinardi, T; Martinelli, A; Trincavelli, L; Tintori, C.
Cytotoxic effects of a novel pyrazolopyrimidine derivative entrapped in liposomes in anaplastic thyroid cancer cells in vitro and in xenograft tumors in vivo 1-gen-2008 M., Celano; Schenone, Silvia; D., Cosco; M., Navarra; E., Puxeddu; L., Racanicchi; Brullo, Chiara; E., Varano; S., Alcaro; E., Ferretti; G., Botta; S., Filetti; M., Fresta; M., Botta; D., Russo
Synthesis, biological evaluation and docking studies of 4-amino substituted 1H-pyrazolo[3,4-d]pyrimidines 1-gen-2008 Schenone, Silvia; Brullo, Chiara; Bruno, Olga; Bondavalli, Francesco; Mosti, Luisa; G., Maga; E., Crespan; F., Carraro; F., Manetti; C., Tintori; M., Botta
Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists: synthesis, biological evaluation, and development of an A1 bovine receptor model. 1-gen-2008 Tuccinardi, T; Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Mosti, Luisa; Zizzari, At; Tintori, C; Manetti, F; Ciampi, O; Trincavelli, Ml; Martini, C; Martinelli, A; Botta, M.
Structure-based optimization of pyrazolo[3,4-d]pyrimidines as Abl inhibitors and antiproliferative agents toward human leukemia cell lines 1-gen-2008 Manetti, F.; Brullo, Chiara; Magnani, M.; Mosci, F.; Chelli, B.; Crespan, E.; Schenone, Silvia; Naldini, A.; Bruno, Olga; Trincavelli, M. L.; Maga, G.; Carraro, F.; Martini, C.; Bondavalli, Francesco; Botta, M.
3D QSAR models built on structure-based alignments of Abl tyrosine kinase inhibitors. 1-gen-2009 F., Falchi; F., Manetti; F., Carraro; A., Naldini; G., Maga; E., Crespan; Schenone, Silvia; Bruno, Olga; Brullo, Chiara; M. Botta, .
New selective phosphodiesterase 4D inhibitors differently acting on long, short, and supershort isoforms 1-gen-2009 Bruno, Olga; A., Romussi; Spallarossa, Andrea; Brullo, Chiara; Schenone, Silvia; Bondavalli, Francesco; N., Vanthuyne; C., Roussel
New selective PDE4D inhibitors able to discriminate between long, short and supershort isoforms 1-gen-2009 Bruno, Olga; Alessia, Romussi; Brullo, Chiara; Schenone, Silvia; Bondavalli, Francesco
Selective PDE4D3 inhibitors as potential drugs in memory impairments 1-gen-2009 Bruno, Olga; Romussi, A; Brullo, Chiara; Schenone, S; Bondavalli, F.
1-Methyl and 1-(2-hydroxyalkyl)-5-(3-alkyl/cycloalkyl/phenyl/naphthylureido)-1H-pyrazole-4-carboxylic acid ethyl esters as potent human neutrophil chemotaxis inhibitors 1-gen-2009 Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Schenone, Silvia; Spisani, S; Falzarano, Ms; Varani, K; Barocelli, E; Ballabeni, V; Giorgio, C; Tognolini, M.
Synthesis of new 2-phenyl-1-arylcarbamoyl-2,3-dihydro-1h-imidazo[1,2-b]pyrazoles 7-substituted as potential neutrophil chemotaxis inhibitors 1-gen-2010 Brullo, Chiara; Bruno, Olga; Schenone, Silvia; Bondavalli, Francesco; S., Spisani; K., Varani
Synthesis of new pyrazolo[3,4-d]pyrimidine derivatives as dual src/abl inhibitors 1-gen-2010 Schenone, Silvia; Musumeci, Francesca; Brullo, Chiara; Bondavalli, Francesco; M., Radi; M., Botta
A1 receptors ligands: past, present and future trends. 1-gen-2010 Schenone, Silvia; Brullo, Chiara; Musumeci, Francesca; Bruno, Olga; Botta, M.
Novel dual Src/Abl inhibitors for hematologic and solid malignancies. 1-gen-2010 Schenone, Silvia; Brullo, Chiara; Musumeci, Francesca; Botta, M.
Gebr-7b, a novel selective PDE4D inhibitor, increases beta amyloid secretion in neuronal cultured cells and improves cognitive function in rodents 1-gen-2010 Ricciarelli, Roberta; Fedele, Ernesto; J., PRICKAERTS J; Brullo, Chiara; Balbi, Alessandro; Canepa, Elisa; A., Cavallero; E., Bollen; Marinari, Umberto; Pronzato, MARIA ADELAIDE; Domenicotti, CINZIA MARIA; Bruno, Olga
Synthesis of new pyrazolo[3,4-d]pyrimidines 6-alkyl substituted Bcr-Abl tyrosine kinase inhibitors 1-gen-2010 Musumeci, F.; Schenone, S.; Brullo, C.; Bruno, O.; Botta, M.
Hit identification and biological evaluation of anticancer pyrazolopyrimidines endowed with anti-inflammatory activity 1-gen-2010 S., Alcaro; A., Artes; M., Botta; A., Zizzarri; F., Orallo; F., Ortuso; Schenone, Silvia; Brullo, Chiara; M. Y., Cez
Mostrati risultati da 41 a 60 di 171
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