Sfoglia per Autore
Sinthesis in vitro inhibitory activity on human platelet aggregation of novel properly substituted 4-(1-piperazinyl)-coumarins
2004-01-01 DI BRACCIO, M; Grossi, G; Roma, G; Signorello, M.; Leoncini, G
Mechanisms involved in the antiplatelet activity of 8-methyl-4-(1-piperazinyl)-7-(3-pyridinylmethoxy)-2H-1-benzopyran-2-one (RC414)
2004-01-01 Leoncini, Giuliana; Signorello, MARIA GRAZIA; D., Bruzzese; DI BRACCIO, Mario; Grossi, Giancarlo; Roma, Giorgio
1,5-Benzodiazepines XIV. Synthesis of new substituted 9H-bis[1,2,4]triazolo[4,3-a:3',4'-d][1,5]benzodiazepines and related compounds endowed with in vitro cytotoxic properties
2005-01-01 DI BRACCIO, Mario; Grossi, Giancarlo; Ceruti, M.; Rocco, F.; Loddo, R.; Sanna, G.; Busonera, B.; Marreddu, M.; Marongiu, M. E.
1,8-Naphthyridines V.Novel N-substituted 5-amino-N,N-diethyl-9-isopropyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, as potent anti-inflammatory and/or analgesic agents completely devoid of acute gastrolesivity
2005-01-01 Grossi, Giancarlo; DI BRACCIO, Mario; Roma, Giorgio; Ballabeni, V.; Tognolini, M.; Barocelli, E.
Synthesis and in vitro antiplatelet activity of new 4-(1-piperazinyl)coumarin derivatives. Human platelet phosphodiesterase 3 inhibitory properties of the two most effective compounds described and molecular modeling study on their interactions with phosphodiesterase 3A catalytic site
2007-01-01 Roma, Giorgio; DI BRACCIO, Mario; Grossi, Giancarlo; Piras, D.; Leoncini, Giuliana; Bruzzese, D.; Signorello, MARIA GRAZIA; Fossa, Paola; Mosti, Luisa
1,8-Naphthyridines VI. Synthesis and anti-inflammatory activity of 5-(alkylamino)-N,N-diethyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6 carboxamides with a new substitution pattern on the triazole ring
2008-01-01 DI BRACCIO, Mario; Grossi, Giancarlo; Roma, Giorgio; D., Piras; Mattioli, Francesca; Gosmar, Marzia
1,8-Naphthyridines VII. New substituted 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides and their isosteric analogues, exhibiting notable anti-inflammatory and/or analgesic activities, but no acute gastrolesivity
2008-01-01 Roma, Giorgio; Grossi, Giancarlo; DI BRACCIO, Mario; Piras, D.; Ballabeni, V.; Tognolini, M.; Bertoni, S.; Barocelli, E.
Efficient one-pot synthesis of N-substituted 2-aminochromones, their benzo-fused derivatives, and diaminobenzodipyrandiones of two new structural classes
2010-01-01 Giorgio, Roma; Daniela, Piras; DI BRACCIO, Mario; Grossi, Giancarlo
New 1,5 - Benzodiazepine Compounds: Activity at Native GABAA Receptors
2010-01-01 Gatta, Elena; A., Cupello; DI BRACCIO, Mario; Grossi, Giancarlo; R., Ferruzzi; Roma, Giorgio; Robello, Mauro
1,8-Naphthyridines VIII. Novel 5-aminoimidazo[1,2-a][1,8]naphthyridine-6-carboxamide and 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamide derivatives showing potent analgesic or anti-inflammatory activity, respectively, and completely devoid of acute gastrolesivity.
2010-01-01 Giorgio, Roma; DI BRACCIO, Mario; Grossi, Giancarlo; Daniela, Piras; Vigilio, Ballabeni; Massimiliano, Tognolini; Simona, Bertoni; Elisabetta, Barocelli
Fine molecular tuning at position 4 of 2H-chromen-2-one derivatives in the search of potent and selective monoamine oxidase B inhibitors
2013-01-01 Leonardo, Pisani; Marco, Catto; Orazio, Nicolotti; Grossi, Giancarlo; Mario Di, Braccio; Ramon Soto, Otero; Estefania Mendez, Alvarez; Angela, Stefanachi; Domenico, Gadaleta; Angelo, Carotti
GABA A Receptors of Cerebellar Granule in Culture: Interaction with Benzodiazepines
2013-01-01 Cupello, Aroldo; Mario Di, Braccio; Gatta, Elena; Grossi, Giancarlo; Nikas, Periklis; Pellistri, Francesca; Robello, Mauro
Modulation of native GABAA receptor activity by triazolo 1,5-benzodiazepines
2013-01-01 Nikas, Periklis; Gatta, Elena; A., Cupello; DI BRACCIO, Mario; Grossi, Giancarlo; Pellistri, Francesca; Robello, Mauro
Synthesis, in vitro antiplatelet activity and molecular modelling studies of 10-substituted 2-(1-piperazinyl)pyrimido[1,2-a]benzimidazol-4(10H)-ones
2013-01-01 DI BRACCIO, Mario; Grossi, Giancarlo; Signorello, MARIA GRAZIA; Leoncini, Giuliana; Cichero, Elena; Fossa, Paola; Alfei, Silvana; Damonte, Gianluca
1,8-Naphthyridines IX. Potent anti-inflammatory and/or analgesic activity of a new group of substituted 5-amino[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides, of some their Mannich base derivatives and of one novel substituted 5-amino-10-oxo-10Hpyrimido[ 1,2-a][1,8]naphthyridine-6-carboxamide derivative
2014-01-01 Mario Di Braccio, A; Grossi, Giancarlo; Alfei, Silvana; Vigilio Ballabeni, C; Massimiliano Tognolini, C; Lisa Flammini, C; Carmine Giorgio, C; Simona Bertoni, C; Elisabetta Barocelli, C.
Study of the Interaction of 1,4- and 1,5-Benzodiazepines with GABAA Receptors of Rat Cerebellum Granule Cells in Culture
2015-01-01 Nikas, Periklis; Gatta, Elena; Cupello, Aroldo; DI BRACCIO, Mario; Grossi, Giancarlo; Pellistri, Francesca; Robello, Mauro
Analogs, formulations and derivatives of imatinib: A patent review
2015-01-01 Musumeci, Francesca; Schenone, Silvia; Grossi, Giancarlo; Brullo, Chiara; Sanna, Monica
Anticonvulsive Activity in Audiogenic DBA/2 Mice of 1,4-Benzodiazepines and 1,5-Benzodiazepines with Different Activities at Cerebellar Granule Cell GABAA Receptors
2016-01-01 Gatta, Elena; Cupello, Aroldo; DI BRACCIO, Mario; Grossi, Giancarlo; Robello, Mauro; Scicchitano, Francesca; Russo, Emilio; De Sarro, Giovambattista
Pyrrolo[2,3-d]pyrimidines as kinase inhibitors
2017-01-01 Musumeci, Francesca; Sanna, Monica; Grossi, Giancarlo; Brullo, Chiara; Fallacara, Anna Lucia; Schenone, Silvia
Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma
2017-01-01 Musumeci, F; Fallacara, Al; Brullo, C; Grossi, G; Botta, L; Calandro, P; Chiariello, M; Kissova, M; Crespan, E; Maga, G; Schenone, S.
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