ZOPPI, VITTORIA

ZOPPI, VITTORIA  

100019 - Dipartimento di chimica e chimica industriale  

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Titolo Data di pubblicazione Autore(i) File
BRD9-targeting PROTACs: design, synthesis and biological evaluation 1-gen-2018 Zoppi, V; Testa, A; Maniaci, C; Hughes, S; Spallarossa, A; Ciulli, A
Hydrophilic and amphiphilic water-soluble dendrimer prodrugs suitable for parenteral administration of a non-soluble non-nucleoside HIV-1 reverse transcriptase inhibitor thiocarbamate derivative 1-gen-2018 Alfei, Silvana; Catena, Silvia; Ponassi, Marco; Rosano, Camillo; Zoppi, Vittoria; Spallarossa, Andrea
Iterative design and optimization of initially inactive Proteolysis Targeting Chimeras (PROTACs) identify VZ185 as a potent, fast and selective von Hippel-Lindau (VHL)-based dual degrader probe of BRD9 and BRD7 1-gen-2019 Zoppi, Vittoria; J Hughes, Scott; Maniaci, Chiara; Testa, Andrea; Gmaschitz, Teresa; Wieshofer, Corinna; Koegl, Manfred; Riching, Kristin; Daniels, Danette L.; Spallarossa, Andrea; Ciulli, Alessio
Studies on Proteolysis Targeting Chimeras: platform technology for targeted protein degradation in drug discovery 11-mar-2019 Zoppi, Vittoria
Synthesis and SAR studies of novel merbarone analogues 1-gen-2016 Zoppi, Vittoria; Odone, A; Ponassi, M; Rosano, C; Spallarossa, A