Sfoglia per Autore
Antitubercular and antiprotozoal activities of quinolizidinyl/pyrrolizidinylalkyliminophenazines
2012-01-01 Novelli, Federica; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Anna, Sparatore; Paola, Molicotti; Stefania, Zanetti
Celecoxib, a COX-2 inhibitor, blocks microglial activation induced by a neurotoxic conformer of hPrP90-231
2012-01-01 Villa, Valentina; Corsaro, Alessandro; THELLUNG DE COURTELARY, Stefano; Tonelli, Michele; Tasso, Bruno; Sparatore, Fabio; Silvia, Leone; Fucile, Carmen; Florio, Tullio
CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation
2013-01-01 M., Sala; D., Braida; L., Pucci; I., Manfredi; M. J., Marks; C. R., Wageman; S. R., Grady; B., Loi; S., Fucile; F., Fasoli; M., Zoli; Tasso, Bruno; Sparatore, Fabio; F., Clementi; C., Gotti
(+)-Laburnamine, a natural selective ligand and partial agonist for the α4β2 nicotinic receptor subtype
2013-01-01 Tasso, Bruno; Novelli, Federica; Sparatore, Fabio; F., Casoli; C., Gotti
Primary anti-proliferative activity evaluation of 1-(quinolizidin-1'-yl)methyl- and 1-([Formula: see text]-tert-amino)alkyl-substituted 2-phenyl-, 2-benzyl- and 2-[(benzotriazol-1/2-yl)methyl]benzimidazoles on human cancer cell lines.
2013-01-01 Tonelli, Michele; Tasso, Bruno; Lorenzo, Mina; Giuseppe, Paglietti; Boido, Vito; Sparatore, Fabio
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents
2014-01-01 Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta
On the self-condensation of aminoguanidine leading to 1,1,4,10,10-pentaamino-2,3,5,6,8,9-hexaazadeca-1,3,5,7,9-pentaene (Structure elucidation through X-ray powder diffraction)
2014-01-01 Tasso, Bruno; G., Pirisino; Novelli, Federica; D., Garzon; R., Fruttero; Sparatore, Fabio; V., Colombo; A., Sironi
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines
2014-01-01 Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Anna, Sparatore; Boido, Vito; Sparatore, Fabio; Sara, Cannas; Paola, Molicotti; Stefania, Zanetti; Silvia, Parapini; Roberta, Loddo
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5
2015-01-01 Roberta, Loddo; Novelli, Federica; Anna, Sparatore; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Gabriella, Collu; Ilenia, Delogu; Gabriele, Giliberti; Paolo, La Colla
Multitarget Therapeutic Leads for Alzheimer’s Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and beta-Amyloid (Abeta) Aggregation
2015-01-01 Tonelli, Michele; Catto, Marco*; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Iusco, Giovanna; Pisani, Leonardo; De Stradis, Angelo; Denora, Nunzio; Sparatore, Anna; Boido, Vito; Carotti, Angelo; Sparatore, Fabio
Clofazimine analogs with antileishmanial and antiplasmodial activity
2015-01-01 Barteselli, A.; Casagrande, M.; Basilico, N.; Parapini, S.; Rusconi, C. M.; Tonelli, Michele; Boido, Vito; Taramelli, D.; Sparatore, Fabio; Sparatore, A.
Synthesis and antiplasmodial activity of novel chloroquine analogues with bulky basic side chains
2015-01-01 Tasso, Bruno; Novelli, Federica; Tonelli, Michele; Barteselli, Anna; Basilico, Nicoletta; Parapini, Silvia; Taramelli, Donatella; Sparatore, Anna; Sparatore, Fabio
New arylsparteine derivatives as positive inotropic drugs
2017-01-01 Boido, Vito; Ercoli, Marcella; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Sparatore, Fabio; Cichero, Elena; Fossa, Paola; Dorigo, Paola; Froldi, Guglielmina
Benzimidazole derivatives endowed with potent antileishmanial activity
2018-01-01 Tonelli, Michele; Gabriele, Elena; Piazza, Francesca; Basilico, Nicoletta; Parapini, Silvia; Tasso, Bruno; Loddo, Roberta; Sparatore, Fabio; Sparatore, Anna
Quinolizidine-derived lucanthone and amitriptyline analogues endowed with potent antileishmanial activity
2020-01-01 Tonelli, M.; Sparatore, A.; Basilico, N.; Cavicchini, L.; Parapini, S.; Tasso, B.; Laurini, E.; Pricl, S.; Boido, V.; Sparatore, F.
Optimization of the clofazimine structure leads to a highly water-soluble C3-aminopyridinyl riminophenazine endowed with improved anti-Wnt and anti-cancer activity in vitro and in vivo
2021-01-01 Koval, A.; Bassanini, I.; Xu, J.; Tonelli, M.; Boido, V.; Sparatore, F.; Amant, F.; Annibali, D.; Leucci, E.; Sparatore, A.; Katanaev, V. L.
Further quinolizidine derivatives as antiarrhythmic agents-3
2023-01-01 Tasso, Bruno; Beatrice Mattioli, Laura; Tonelli, Michele; Boido, Vito; Chiarini, Alberto; Sparatore, Fabio; Budriesi, Roberta
Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease
2023-01-01 Tonelli, Michele; Catto, Marco; Sabaté, Raimon; Francesconi, Valeria; Laurini, Erik; Pricl, Sabrina; Pisani, Leonardo; Valeria Miniero, Daniela; Maria Liuzzi, Grazia; Gatta, Elena; Relini, Annalisa; Gavín, Rosalina; Antonio Del Rio, Jose; Sparatore, Fabio; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Antitubercular and antiprotozoal activities of quinolizidinyl/pyrrolizidinylalkyliminophenazines | 1-gen-2012 | Novelli, Federica; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Anna, Sparatore; Paola, Molicotti; Stefania, Zanetti | |
Celecoxib, a COX-2 inhibitor, blocks microglial activation induced by a neurotoxic conformer of hPrP90-231 | 1-gen-2012 | Villa, Valentina; Corsaro, Alessandro; THELLUNG DE COURTELARY, Stefano; Tonelli, Michele; Tasso, Bruno; Sparatore, Fabio; Silvia, Leone; Fucile, Carmen; Florio, Tullio | |
CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation | 1-gen-2013 | M., Sala; D., Braida; L., Pucci; I., Manfredi; M. J., Marks; C. R., Wageman; S. R., Grady; B., Loi; S., Fucile; F., Fasoli; M., Zoli; Tasso, Bruno; Sparatore, Fabio; F., Clementi; C., Gotti | |
(+)-Laburnamine, a natural selective ligand and partial agonist for the α4β2 nicotinic receptor subtype | 1-gen-2013 | Tasso, Bruno; Novelli, Federica; Sparatore, Fabio; F., Casoli; C., Gotti | |
Primary anti-proliferative activity evaluation of 1-(quinolizidin-1'-yl)methyl- and 1-([Formula: see text]-tert-amino)alkyl-substituted 2-phenyl-, 2-benzyl- and 2-[(benzotriazol-1/2-yl)methyl]benzimidazoles on human cancer cell lines. | 1-gen-2013 | Tonelli, Michele; Tasso, Bruno; Lorenzo, Mina; Giuseppe, Paglietti; Boido, Vito; Sparatore, Fabio | |
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents | 1-gen-2014 | Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta | |
On the self-condensation of aminoguanidine leading to 1,1,4,10,10-pentaamino-2,3,5,6,8,9-hexaazadeca-1,3,5,7,9-pentaene (Structure elucidation through X-ray powder diffraction) | 1-gen-2014 | Tasso, Bruno; G., Pirisino; Novelli, Federica; D., Garzon; R., Fruttero; Sparatore, Fabio; V., Colombo; A., Sironi | |
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines | 1-gen-2014 | Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Anna, Sparatore; Boido, Vito; Sparatore, Fabio; Sara, Cannas; Paola, Molicotti; Stefania, Zanetti; Silvia, Parapini; Roberta, Loddo | |
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5 | 1-gen-2015 | Roberta, Loddo; Novelli, Federica; Anna, Sparatore; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Gabriella, Collu; Ilenia, Delogu; Gabriele, Giliberti; Paolo, La Colla | |
Multitarget Therapeutic Leads for Alzheimer’s Disease: Quinolizidinyl Derivatives of Bi- and Tricyclic Systems as Dual Inhibitors of Cholinesterases and beta-Amyloid (Abeta) Aggregation | 1-gen-2015 | Tonelli, Michele; Catto, Marco*; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Iusco, Giovanna; Pisani, Leonardo; De Stradis, Angelo; Denora, Nunzio; Sparatore, Anna; Boido, Vito; Carotti, Angelo; Sparatore, Fabio | |
Clofazimine analogs with antileishmanial and antiplasmodial activity | 1-gen-2015 | Barteselli, A.; Casagrande, M.; Basilico, N.; Parapini, S.; Rusconi, C. M.; Tonelli, Michele; Boido, Vito; Taramelli, D.; Sparatore, Fabio; Sparatore, A. | |
Synthesis and antiplasmodial activity of novel chloroquine analogues with bulky basic side chains | 1-gen-2015 | Tasso, Bruno; Novelli, Federica; Tonelli, Michele; Barteselli, Anna; Basilico, Nicoletta; Parapini, Silvia; Taramelli, Donatella; Sparatore, Anna; Sparatore, Fabio | |
New arylsparteine derivatives as positive inotropic drugs | 1-gen-2017 | Boido, Vito; Ercoli, Marcella; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Sparatore, Fabio; Cichero, Elena; Fossa, Paola; Dorigo, Paola; Froldi, Guglielmina | |
Benzimidazole derivatives endowed with potent antileishmanial activity | 1-gen-2018 | Tonelli, Michele; Gabriele, Elena; Piazza, Francesca; Basilico, Nicoletta; Parapini, Silvia; Tasso, Bruno; Loddo, Roberta; Sparatore, Fabio; Sparatore, Anna | |
Quinolizidine-derived lucanthone and amitriptyline analogues endowed with potent antileishmanial activity | 1-gen-2020 | Tonelli, M.; Sparatore, A.; Basilico, N.; Cavicchini, L.; Parapini, S.; Tasso, B.; Laurini, E.; Pricl, S.; Boido, V.; Sparatore, F. | |
Optimization of the clofazimine structure leads to a highly water-soluble C3-aminopyridinyl riminophenazine endowed with improved anti-Wnt and anti-cancer activity in vitro and in vivo | 1-gen-2021 | Koval, A.; Bassanini, I.; Xu, J.; Tonelli, M.; Boido, V.; Sparatore, F.; Amant, F.; Annibali, D.; Leucci, E.; Sparatore, A.; Katanaev, V. L. | |
Further quinolizidine derivatives as antiarrhythmic agents-3 | 1-gen-2023 | Tasso, Bruno; Beatrice Mattioli, Laura; Tonelli, Michele; Boido, Vito; Chiarini, Alberto; Sparatore, Fabio; Budriesi, Roberta | |
Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease | 1-gen-2023 | Tonelli, Michele; Catto, Marco; Sabaté, Raimon; Francesconi, Valeria; Laurini, Erik; Pricl, Sabrina; Pisani, Leonardo; Valeria Miniero, Daniela; Maria Liuzzi, Grazia; Gatta, Elena; Relini, Annalisa; Gavín, Rosalina; Antonio Del Rio, Jose; Sparatore, Fabio; Carotti, Angelo |
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