CESARINI, SARA
CESARINI, SARA
58 - Dipartimento di Scienze farmaceutiche (attivo dal 01/01/1997 al 18/07/2012)
(Hetero)aroyl esters of 2-(N-phthalimido)ethanol and analogues: parallel synthesis, anti-HIV-1 activity and cytotoxicity
2010-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Schenone, Silvia; LA COLLA, P; Collu, G; Sanna, G; Loddo, R.
6-amino-4-oxo-1,3-diphenyl-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl derivatives as a new class of potent inhibitors of Interleukin-8-induced neutrophil chemotaxis
2009-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Bruno, Olga; Arduino, N; Bertolotto, M; Dallegri, Franco; Tognolini, M; Gobbetti, T; Barocelli, E.
A novel potent non-nucleoside reverse transcriptase inhibitor acylthiocarbamate derivative with extensive intramolecular pi-pi interactions
2006-01-01 Mugnoli, A; Borassi, A; Spallarossa, Andrea; Cesarini, Sara
A Successful Application of Parallel Synthesis to Computer-Assisted Structural Optimization of New Leads Targeting Human Immunodeficiency Virus-1 Reverse Transcriptase. The Case of Acylthiocarbamates and Thiocarbamates
2008-01-01 Ranise, Angelo; Spallarossa, Andrea; Cesarini, Sara
Acylthiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors: docking studies and ligand-based CoMFA and CoMSIA analyses
2009-01-01 Cichero, Elena; Cesarini, Sara; Spallarossa, Andrea; Mosti, Luisa; Fossa, Paola
CoMFA and CoMSIA analyses on 1,2,3,4-tetrahydropyrrolo[3,4-b]indole and benzimidazole derivatives as selective CB2 receptor agonists.
2010-01-01 Cichero, Elena; Cesarini, Sara; Mosti, Luisa; Fossa, Paola
CoMFA and CoMSIA analyses on 4-oxo-1,4-dihydroquinoline and 4-oxo-1,4-dihydro-1,5-, -1,6- and -1,8-naphthyridine derivatives as selective CB2 receptor agonists
2010-01-01 Cichero, Elena; Cesarini, Sara; Mosti, Luisa; Fossa, Paola
Computational studies of the binding mode and 3D-QSAR analyses of symmetric formimidoester disulfides: a new class of non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Cichero, Elena; Cesarini, Sara; Spallarossa, Andrea; Mosti, Luisa; Fossa, Paola
Crystal structures of HIV-1 reverse transcriptase in complexes with thiocarbamate non-nucleoside inhibitors
2008-01-01 Spallarossa, Andrea; Cesarini, Sara; Ranise, Angelo; Ponassi, M; Unge, T; Bolognesi, M.
N-acylated and N,N'-diacylated imidazolidine-2-thione derivatives and N,N'-diacylated tetrahydropyrimidine-2(1H)-thione analogues: synthesis and antiproliferative activity.
2009-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Schenone, Silvia; Rosano, C; LA COLLA, P; Sanna, G; Busonera, B; Loddo, R.
Non-receptor tyrosine kinase Fes as a target in oncology
2008-01-01 Zaborowska, J; Spallarossa, Andrea; Ranise, Angelo; Cesarini, Sara; Stec, E; Condorelli, F; Rosano, C.
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2008-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Schenone, Silvia; Bruno, Olga; LA COLLA, P.; Casula, L.; Collu, G.; Sanna, G.; Loddo, R.
Parallel synthesis of O-phenoxyethyl and O-adamantyl N-acyl thiocarbamates endowed with antiproliferative activity.
2009-01-01 Spallarossa, Andrea; Cesarini, Sara; Schenone, Silvia; Ranise, Angelo
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, Andrea; Cesarini, Sara; Ranise, Angelo; Schenone, Silvia; Bruno, Olga; A., Borassi; P., La Colla; M., Pezzullo; G., Sanna; G., Collu; B., Secci; R., Loddo
Structure-based Design, Parallel Synthesis, SAR and Molecular Modelling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea (PETT) Derivatives.
2005-01-01 Ranise, Angelo; Spallarossa, Andrea; Cesarini, Sara; Bondavalli, Francesco; Schenone, Silvia; Bruno, Olga; Menozzi, Giulia; Fossa, Paola; Mosti, Luisa; M., LA COLLA; G., Sanna; M., Murreddu; G., Collu; B., Busonera; M. E., Marongiu; A., Pani; P., LA COLLA; R., Loddo
Synthesis of indole imminun salts as key-intermediates in a convergent multi-step one-pot stereoselective synthesis of new potent antiproliferative Knoevenagel-type agent
2008-01-01 Caviglia, M; Cesarini, Sara; Spallarossa, Andrea; Fossa, Paola; Mosti, Luisa; Ranise, Angelo
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates
2008-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Fossa, Paola; LA COLLA, P; Sanna, G; Collu, G; Loddo, R.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate
2008-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Bruno, Olga; LA COLLA, P; Secci, B; Collu, G; Loddo, R.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors: docking-based CoMFA and CoMSIA analyses
2009-01-01 Cichero, Elena; Cesarini, Sara; Fossa, Paola; Spallarossa, Andrea; Mosti, Luisa
Unprecedented one-pot stereoselective synthesis of Knoevenagel-type derivatives via in situ condensation of N-methyleniminium salts of ethylenethiourea and ethyleneurea with active methylene reagents
2007-01-01 Ranise, Angelo; Cesarini, Sara; Spallarossa, Andrea; Sancassan, F.; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Menozzi, Giulia; Fossa, Paola; Mosti, Luisa