Sfoglia per Autore
New milrinone analogues:in vitro study of structure-activity relationships for positive inotropic effect, antagonism towards endogenous adenosine and inhibition of cardiac type III phosphodiesterase
2003-01-01 Floreani, M.; Fossa, Paola; Gessi, S.; Mosti, Luisa; Borea, P. A.; Dorigo, P.
4-Substituted 1,5-diarylpyrazoles, analogues of celecoxib: synthesis and preliminary evaluation of biological properties
2003-01-01 Menozzi, Giulia; Merello, L.; Fossa, Paola; Mosti, Luisa; Piana, A.; Mattioli, Francesca
Exploring the molecular basis of selectivity in A1 adenosine receptors antagonist: a case study
2003-01-01 Giordanetto, F.; Fossa, Paola; Menozzi, Giulia; Schenone, Silvia; Bondavalli, Francesco; Ranise, Angelo; Mosti, Luisa
In silico rationalization of the structural and physicochemical requirements for photobiological activity in angelicine derivatives and their heteroanalogues
2003-01-01 Giordanetto, F.; Fossa, Paola; Menozzi, Giulia; Mosti, Luisa
Synthesis of N-substituted-N-acylthioureas of 4-substituted piperazines endowed with local anaesthetic, antihyperlipidemic, antiproliferative activities and antiarrythmic, analgesic, antiaggregating actions
2003-01-01 Ranise, Angelo; Spallarossa, Andrea; Bruno, Olga; Schenone, Silvia; Fossa, Paola; Menozzi, Giulia; Bondavalli, Francesco; Mosti, Luisa; Capuano, A.; Mazzeo, F.; Falcone, G.; Filippelli, W.
Antiproliferative activity of new 1-aryl-4-amino-1H-pyrazolo[3,4-d]pyrimidine derivatives toward the human epidermoid carcinoma A431 cell line
2004-01-01 Schenone, Silvia; Bruno, Olga; Bondavalli, Francesco; Ranise, Angelo; Mosti, Luisa; Menozzi, Giulia; Fossa, Paola; Donnini, S.; Santoro, A.; Ziche, M.; Manetti, F.; Botta, M.
Synthesis, antimicrobial activity and molecular modelling studies of halogenated 4-[1H-imidazol-1-yl(phenyl)methyl]-1,5-diphenyl-1H-pyrazoles
2004-01-01 Menozzi, Giulia; Merello, L.; Fossa, Paola; Schenone, Silvia; Ranise, Angelo; Mosti, Luisa; Bondavalli, Francesco; Loddo, R.; Murgioni, C.; Mascia, V.; LA COLLA, P.; Tamburini, E.
Synthesis of 1-(2-chloro-2-phenylethyl)-6-methylthio-1-H-pyrazolo[3,4-d]pyrimidines 4-amino substituted and their biological evaluation
2004-01-01 Schenone, S.; Bruno, O.; Bondavalli, F.; Ranise, A.; Mosti, L.; Menozzi, G.; Fossa, P.; Manetti, F.; Morbidelli, L.; Trincavelli, L.; Martini, C.; Lucacchini, A.
New pyrazolo[3,4-d]pyrimidines endowed with A431 antiproliferative activity and inhibitory properties of Src phosphorylation
2004-01-01 Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Brullo, Chiara; Fossa, Paola; Mosti, Luisa; Menozzi, Giulia; Carraro, F.; Naldini, A.; Bernini, C.; Manetti, F.; Botta, M.
Pyrazolo[3,4-d]pyrimidines endowed with antiproliferative activity on ductal infiltrating carcinoma cells
2004-01-01 F., Carraro; A., Pucci; A., Naldini; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Brullo, Chiara; Fossa, Paola; Menozzi, Giulia; Mosti, Luisa; F., Manetti; M., Botta
Synthesis, Biological Evaluation and Molecular Modeling Studies on Benzothiadiazine Derivatives as PDE4 Selective Inhibitors
2005-01-01 Tait, A.; Luppi, A.; Hatzelmann, A.; Fossa, Paola; Mosti, Luisa
New halogenated 4-aminopyrazolo[3,4-b]pyridines A1 adenosine receptor ligands
2005-01-01 Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Ranise, Angelo; Mosti, Luisa; Menozzi, Giulia; Fossa, Paola; Trincavelli, M. L.; Martini, C.
Insights into Structure-Activity Relationships from Lipophilicity Profiles of Pyridin-2(1H)-one Analogs of the Cardiotonic Agent Milrinone
2005-01-01 DE CANDIA, M.; Fossa, Paola; Cellamare, S.; Mosti, Luisa; Carotti, A.; Altomare, C.
A chemometric approach to predict A1 agonist effect of adenosine analogues
2005-01-01 Fossa, Paola; Mosti, Luisa; Bondavalli, Francesco; Schenone, Silvia; Ranise, Angelo; Casolino, MARIA CHIARA; Forina, Michele
Synthesis and 3D QSAR of new pyrazolo[3,4-b]pyridines: potent and selective inhibitors of A1 adenosine receptors
2005-01-01 F., Manetti; Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Ranise, Angelo; Mosti, Luisa; Menozzi, Giulia; Fossa, Paola; M. L., Trincavelli; C., Martini; A., Martinelli; C., Tintori; M., Botta
Structure-based Design, Parallel Synthesis, SAR and Molecular Modelling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea (PETT) Derivatives.
2005-01-01 Ranise, Angelo; Spallarossa, Andrea; Cesarini, Sara; Bondavalli, Francesco; Schenone, Silvia; Bruno, Olga; Menozzi, Giulia; Fossa, Paola; Mosti, Luisa; M., LA COLLA; G., Sanna; M., Murreddu; G., Collu; B., Busonera; M. E., Marongiu; A., Pani; P., LA COLLA; R., Loddo
New pyrazolo[3,4-b]pyridones as selective A1 adenosine receptor antagonists: synthesis, biological evaluation and molecular modeling studies
2005-01-01 Fossa, Paola; Pestarino, M; Menozzi, Giulia; Mosti, Luisa; Schenone, Silvia; Ranise, Angelo; Bondavalli, Francesco; Trincavelli, Ml; Lucacchini, A; Martini, C.
Synthesis of pyrazolo[3,4-d]pyridines selective antagonists of A1 adenosine receptors
2006-01-01 Schenone, Silvia; Brullo, Chiara; Ranise, Angelo; Bondavalli, Francesco; Mosti, Luisa; Fossa, Paola; Menozzi, Giulia; Trincavelli, L; Martini, C; Manetti, F; Tintori, C; Botta, M.
Pyrazolo[3,4-d]pyrimidines as potent antiproliferative and proapoptotic agents toward A431 and 8701-BC cells in culture via inhibition of c-Src phosphorylation
2006-01-01 Carraro, F; Naldini, A; Pucci, A; Locatelli, G. A.; Maga, ; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Brullo, Chiara; Fossa, Paola; Menozzi, Giulia; Mosti, Luisa; Modugno, M; Tintori, C; Manetti, F; Botta, M.
Synthesis of new pyrazolo[3,4-b]pyridines: new selective A1 adenosine receptor antagonists
2006-01-01 Brullo, Chiara; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Mosti, Luisa; Trincavelli, M. L.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
New milrinone analogues:in vitro study of structure-activity relationships for positive inotropic effect, antagonism towards endogenous adenosine and inhibition of cardiac type III phosphodiesterase | 1-gen-2003 | Floreani, M.; Fossa, Paola; Gessi, S.; Mosti, Luisa; Borea, P. A.; Dorigo, P. | |
4-Substituted 1,5-diarylpyrazoles, analogues of celecoxib: synthesis and preliminary evaluation of biological properties | 1-gen-2003 | Menozzi, Giulia; Merello, L.; Fossa, Paola; Mosti, Luisa; Piana, A.; Mattioli, Francesca | |
Exploring the molecular basis of selectivity in A1 adenosine receptors antagonist: a case study | 1-gen-2003 | Giordanetto, F.; Fossa, Paola; Menozzi, Giulia; Schenone, Silvia; Bondavalli, Francesco; Ranise, Angelo; Mosti, Luisa | |
In silico rationalization of the structural and physicochemical requirements for photobiological activity in angelicine derivatives and their heteroanalogues | 1-gen-2003 | Giordanetto, F.; Fossa, Paola; Menozzi, Giulia; Mosti, Luisa | |
Synthesis of N-substituted-N-acylthioureas of 4-substituted piperazines endowed with local anaesthetic, antihyperlipidemic, antiproliferative activities and antiarrythmic, analgesic, antiaggregating actions | 1-gen-2003 | Ranise, Angelo; Spallarossa, Andrea; Bruno, Olga; Schenone, Silvia; Fossa, Paola; Menozzi, Giulia; Bondavalli, Francesco; Mosti, Luisa; Capuano, A.; Mazzeo, F.; Falcone, G.; Filippelli, W. | |
Antiproliferative activity of new 1-aryl-4-amino-1H-pyrazolo[3,4-d]pyrimidine derivatives toward the human epidermoid carcinoma A431 cell line | 1-gen-2004 | Schenone, Silvia; Bruno, Olga; Bondavalli, Francesco; Ranise, Angelo; Mosti, Luisa; Menozzi, Giulia; Fossa, Paola; Donnini, S.; Santoro, A.; Ziche, M.; Manetti, F.; Botta, M. | |
Synthesis, antimicrobial activity and molecular modelling studies of halogenated 4-[1H-imidazol-1-yl(phenyl)methyl]-1,5-diphenyl-1H-pyrazoles | 1-gen-2004 | Menozzi, Giulia; Merello, L.; Fossa, Paola; Schenone, Silvia; Ranise, Angelo; Mosti, Luisa; Bondavalli, Francesco; Loddo, R.; Murgioni, C.; Mascia, V.; LA COLLA, P.; Tamburini, E. | |
Synthesis of 1-(2-chloro-2-phenylethyl)-6-methylthio-1-H-pyrazolo[3,4-d]pyrimidines 4-amino substituted and their biological evaluation | 1-gen-2004 | Schenone, S.; Bruno, O.; Bondavalli, F.; Ranise, A.; Mosti, L.; Menozzi, G.; Fossa, P.; Manetti, F.; Morbidelli, L.; Trincavelli, L.; Martini, C.; Lucacchini, A. | |
New pyrazolo[3,4-d]pyrimidines endowed with A431 antiproliferative activity and inhibitory properties of Src phosphorylation | 1-gen-2004 | Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Brullo, Chiara; Fossa, Paola; Mosti, Luisa; Menozzi, Giulia; Carraro, F.; Naldini, A.; Bernini, C.; Manetti, F.; Botta, M. | |
Pyrazolo[3,4-d]pyrimidines endowed with antiproliferative activity on ductal infiltrating carcinoma cells | 1-gen-2004 | F., Carraro; A., Pucci; A., Naldini; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Brullo, Chiara; Fossa, Paola; Menozzi, Giulia; Mosti, Luisa; F., Manetti; M., Botta | |
Synthesis, Biological Evaluation and Molecular Modeling Studies on Benzothiadiazine Derivatives as PDE4 Selective Inhibitors | 1-gen-2005 | Tait, A.; Luppi, A.; Hatzelmann, A.; Fossa, Paola; Mosti, Luisa | |
New halogenated 4-aminopyrazolo[3,4-b]pyridines A1 adenosine receptor ligands | 1-gen-2005 | Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Ranise, Angelo; Mosti, Luisa; Menozzi, Giulia; Fossa, Paola; Trincavelli, M. L.; Martini, C. | |
Insights into Structure-Activity Relationships from Lipophilicity Profiles of Pyridin-2(1H)-one Analogs of the Cardiotonic Agent Milrinone | 1-gen-2005 | DE CANDIA, M.; Fossa, Paola; Cellamare, S.; Mosti, Luisa; Carotti, A.; Altomare, C. | |
A chemometric approach to predict A1 agonist effect of adenosine analogues | 1-gen-2005 | Fossa, Paola; Mosti, Luisa; Bondavalli, Francesco; Schenone, Silvia; Ranise, Angelo; Casolino, MARIA CHIARA; Forina, Michele | |
Synthesis and 3D QSAR of new pyrazolo[3,4-b]pyridines: potent and selective inhibitors of A1 adenosine receptors | 1-gen-2005 | F., Manetti; Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Ranise, Angelo; Mosti, Luisa; Menozzi, Giulia; Fossa, Paola; M. L., Trincavelli; C., Martini; A., Martinelli; C., Tintori; M., Botta | |
Structure-based Design, Parallel Synthesis, SAR and Molecular Modelling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea (PETT) Derivatives. | 1-gen-2005 | Ranise, Angelo; Spallarossa, Andrea; Cesarini, Sara; Bondavalli, Francesco; Schenone, Silvia; Bruno, Olga; Menozzi, Giulia; Fossa, Paola; Mosti, Luisa; M., LA COLLA; G., Sanna; M., Murreddu; G., Collu; B., Busonera; M. E., Marongiu; A., Pani; P., LA COLLA; R., Loddo | |
New pyrazolo[3,4-b]pyridones as selective A1 adenosine receptor antagonists: synthesis, biological evaluation and molecular modeling studies | 1-gen-2005 | Fossa, Paola; Pestarino, M; Menozzi, Giulia; Mosti, Luisa; Schenone, Silvia; Ranise, Angelo; Bondavalli, Francesco; Trincavelli, Ml; Lucacchini, A; Martini, C. | |
Synthesis of pyrazolo[3,4-d]pyridines selective antagonists of A1 adenosine receptors | 1-gen-2006 | Schenone, Silvia; Brullo, Chiara; Ranise, Angelo; Bondavalli, Francesco; Mosti, Luisa; Fossa, Paola; Menozzi, Giulia; Trincavelli, L; Martini, C; Manetti, F; Tintori, C; Botta, M. | |
Pyrazolo[3,4-d]pyrimidines as potent antiproliferative and proapoptotic agents toward A431 and 8701-BC cells in culture via inhibition of c-Src phosphorylation | 1-gen-2006 | Carraro, F; Naldini, A; Pucci, A; Locatelli, G. A.; Maga, ; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Brullo, Chiara; Fossa, Paola; Menozzi, Giulia; Mosti, Luisa; Modugno, M; Tintori, C; Manetti, F; Botta, M. | |
Synthesis of new pyrazolo[3,4-b]pyridines: new selective A1 adenosine receptor antagonists | 1-gen-2006 | Brullo, Chiara; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Mosti, Luisa; Trincavelli, M. L. |
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