Sfoglia per Autore
Structure-based Design, Parallel Synthesis, SAR and Molecular Modelling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea (PETT) Derivatives.
2005-01-01 Ranise, Angelo; Spallarossa, Andrea; Cesarini, Sara; Bondavalli, Francesco; Schenone, Silvia; Bruno, Olga; Menozzi, Giulia; Fossa, Paola; Mosti, Luisa; M., LA COLLA; G., Sanna; M., Murreddu; G., Collu; B., Busonera; M. E., Marongiu; A., Pani; P., LA COLLA; R., Loddo
X-ray analysis of HIV-1 reverse transcriptase in complex with thiocarbamates: structure-based design and synthesis of new analogues
2006-01-01 Spallarossa, Andrea; Ranise, Angelo; Cesarini, S; Bolognesi, M; Unge, T.
One-pot Stereoselective Synthesis of Knoevenageltype Derivatives Via Condensation of N-Methyleniminium Salts of Ethylenethiourea and Ethyleneurea with Active Methylene Reagents.
2006-01-01 Spallarossa, Andrea; Cesarini, S; Ranise, Angelo; Sancassan, F; Bondavalli, F; Schenone, Silvia; Bruno, Olga; Menozzi, G; Fossa, Paola; Mosti, L.
A novel potent non-nucleoside reverse transcriptase inhibitor acylthiocarbamate derivative with extensive intramolecular pi-pi interactions
2006-01-01 Mugnoli, A; Borassi, A; Spallarossa, Andrea; Cesarini, Sara
Virtual screening and structure based drug design of new Fes/Fps kinase domain inhibitors.
2007-01-01 Rosano, C; Marra, D; Cesarini, S; Ranise, Angelo; Spallarossa, Andrea
Unprecedented one-pot stereoselective synthesis of Knoevenagel-type derivatives via in situ condensation of N-methyleniminium salts of ethylenethiourea and ethyleneurea with active methylene reagents
2007-01-01 Ranise, Angelo; Cesarini, Sara; Spallarossa, Andrea; Sancassan, F.; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Menozzi, Giulia; Fossa, Paola; Mosti, Luisa
Identification of novel pyrazolo[3,4-d]pyrimidine able to inhibit cell proliferation of a human osteogenic sarcoma in vitro and in a xenograft model in mice
2007-01-01 Manetti, F.; Santucci, A.; Locatelli, G. A.; Maga, G.; Spreafico, A.; Serchi, T.; Orlandini, M.; Bemardini, G.; Caradonna, N. P.; Spallarossa, Andrea; Brullo, Chiara; Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Hoffmann, O.; Bologna, M.; Angelucci, A.; Botta, M.
Synthesis of indole imminun salts as key-intermediates in a convergent multi-step one-pot stereoselective synthesis of new potent antiproliferative Knoevenagel-type agent
2008-01-01 Caviglia, M; Cesarini, Sara; Spallarossa, Andrea; Fossa, Paola; Mosti, Luisa; Ranise, Angelo
5-Substituted derivatives of 6-amino-1,3-diphenyl-2-thioxo-2,3-dihydropyrimidin-4(1H)-one as a new class of potent inhibitors of interleukin 8-induced neutrophil chemotaxis
2008-01-01 Cesarini, S; Spallarossa, Andrea; Ranise, Angelo; Bruno, Olga; Arduino, N; Dallegri, Franco; Barocelli, E.
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents
2008-01-01 Spallarossa, Andrea; Cesarini, S; Rotolo, C; Fossa, Paola; Mosti, L; Ranise, Angelo; Sanna, G; Collu, G; Secci, B; Busonera, B; LA COLLA, P; Loddo, R.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates
2008-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Fossa, Paola; LA COLLA, P; Sanna, G; Collu, G; Loddo, R.
Rational design, synthesis and biological evaluation of new 1,5-diarylpyrazole derivatives as CB1 receptor antagonists, structurally related to rimonabant
2008-01-01 Menozzi, Giulia; Fossa, Paola; Cichero, Elena; Spallarossa, Andrea; Ranise, Angelo; Mosti, Luisa
Reattivita' di accettori di Michael atipici con nucleofili azotati
2008-01-01 Rotolo, C; Cesarini, S; Canepa, E; Spallarossa, Andrea; Ranise, Angelo
Non-receptor tyrosine kinase Fes as a target in oncology
2008-01-01 Zaborowska, J; Spallarossa, Andrea; Ranise, Angelo; Cesarini, Sara; Stec, E; Condorelli, F; Rosano, C.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors: docking-based CoMFA and CoMSIA analyses
2008-01-01 Cichero, E; Cesarini, S; Spallarossa, Andrea; Mosti, L; Fossa, Paola
Exploring the binding features of rimonabant analogues and acyclic CB1 antagonists: docking studies and 3D-QSAR analysis
2008-01-01 Cichero, E; Spallarossa, Andrea; Menozzi, Giulia; Mosti, Luisa; Fossa, Paola
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2008-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Schenone, Silvia; Bruno, Olga; LA COLLA, P.; Casula, L.; Collu, G.; Sanna, G.; Loddo, R.
A Successful Application of Parallel Synthesis to Computer-Assisted Structural Optimization of New Leads Targeting Human Immunodeficiency Virus-1 Reverse Transcriptase. The Case of Acylthiocarbamates and Thiocarbamates
2008-01-01 Ranise, Angelo; Spallarossa, Andrea; Cesarini, Sara
Crystal structures of HIV-1 reverse transcriptase in complexes with thiocarbamate non-nucleoside inhibitors
2008-01-01 Spallarossa, Andrea; Cesarini, Sara; Ranise, Angelo; Ponassi, M; Unge, T; Bolognesi, M.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate
2008-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Bruno, Olga; LA COLLA, P; Secci, B; Collu, G; Loddo, R.
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