TASSO, BRUNO
TASSO, BRUNO
100006 - Dipartimento di Farmacia
(+)-Laburnamine, a natural selective ligand and partial agonist for the α4β2 nicotinic receptor subtype
2013-01-01 Tasso, Bruno; Novelli, Federica; Sparatore, Fabio; F., Casoli; C., Gotti
Acridine derivatives as anti-BVDV agents
2011-01-01 Tonelli, Michele; Vettoretti, G; Tasso, Bruno; Novelli, Federica; Boido, Vito; Sparatore, Fabio; Busonera, B; Ouhtit, A; Farci, P; Blois, S; Giliberti, G; La Colla, P.
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines
2014-01-01 Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Anna, Sparatore; Boido, Vito; Sparatore, Fabio; Sara, Cannas; Paola, Molicotti; Stefania, Zanetti; Silvia, Parapini; Roberta, Loddo
Antiviral activity of benzimidazole derivatives. II Antiviral activity of 2-phenylbenzimidazole derivatives.
2010-01-01 Tonelli, Michele; Simone, M; Tasso, Bruno; Novelli, Federica; Boido, Vito; Sparatore, Fabio; Paglietti, G; Pricl, S; Gilberti, G; Blois, S; Ibba, C; Sanna, G; Loddo, R; LA COLLA, P.
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents
2014-01-01 Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5
2015-01-01 Roberta, Loddo; Novelli, Federica; Anna, Sparatore; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Gabriella, Collu; Ilenia, Delogu; Gabriele, Giliberti; Paolo, La Colla
Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives
2009-01-01 Tonelli, Michele; Vazzana, Iana; Tasso, Bruno; Boido, Vito; Sparatore, Fabio; Fermeglia, M.; Paneni, M. S.; Posocco, P.; Pricl, S.; LA COLLA, P.; Ibba, C.; Secci, B.; Collu, G.; Loddo, R.
Benzimidazole derivatives endowed with potent antileishmanial activity
2018-01-01 Tonelli, Michele; Gabriele, Elena; Piazza, Francesca; Basilico, Nicoletta; Parapini, Silvia; Tasso, Bruno; Loddo, Roberta; Sparatore, Fabio; Sparatore, Anna
Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles
2017-01-01 Cichero, Elena; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Delogu, I; Loddo, R.; Bruno, Olga; Fossa, Paola
BMI-1 inhibition fights cancer chemoresistance by altering redox homeostasis and inducing lipid peroxidation
2023-01-01 Valenti, Ge; Tasso, B; Traverso, N; Monteleone, L; Marengo, B; Domenicotti, C
Btk inhibitors: a medicinal chemistry and drug delivery perspective
2021-01-01 Brullo, C.; Villa, C.; Tasso, B.; Russo, E.; Spallarossa, A.
CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation
2013-01-01 M., Sala; D., Braida; L., Pucci; I., Manfredi; M. J., Marks; C. R., Wageman; S. R., Grady; B., Loi; S., Fucile; F., Fasoli; M., Zoli; Tasso, Bruno; Sparatore, Fabio; F., Clementi; C., Gotti
Celecoxib Inhibits Prion Protein 90-231-Mediated Pro-inflammatory Responses in Microglial Cells
2016-01-01 Villa, Valentina; THELLUNG DE COURTELARY, Stefano; Corsaro, Alessandro; Novelli, Federica; Tasso, Bruno; Colucci D’Amato, L.; Gatta, Elena; Tonelli, Michele; Florio, Tullio
Cytisine derivatives as ligands for neuronal nicotine receptors and with various pharmacological activities
2003-01-01 Canu, Caterina; Tasso, Bruno; Boido, Vito; Sparatore, Fabio
Differential modulation of SIRT6 deacetylase and deacylase activities by lysine-based small molecules
2020-01-01 Sociali, G.; Liessi, N.; Grozio, A.; Caffa, I.; Parenti, M. D.; Ravera, S.; Tasso, B.; Benzi, A.; Nencioni, A.; Del Rio, A.; Robina, I.; Millo, E.; Bruzzone, S.
Discovery of Novel Thiazole-Based SIRT2 Inhibitors as Anticancer Agents: Molecular Modeling, Chemical Synthesis and Biological Assays
2024-01-01 Piacente, F.; Guccione, G.; Scarano, N.; Lunaccio, D.; Miro, C.; Abbotto, E.; Salis, A.; Tasso, B.; Dentice, M.; Bruzzone, S.; Cichero, E.; Millo, E.
Discovery of novel VX-809 hybrid derivatives as F508del-CFTR correctors by molecular modeling, chemical synthesis and biological assays
2020-01-01 Parodi, A.; Righetti, G.; Pesce, E.; Salis, A.; Tasso, B.; Urbinati, C.; Tomati, V.; Damonte, G.; Rusnati, M.; Pedemonte, N.; Cichero, E.; Millo, E.
Efficacy of novel acridine derivatives in the inhibition of hPrP90-231 prion protein fragment toxicity
2011-01-01 Villa, Valentina; Tonelli, Michele; THELLUNG DE COURTELARY, Stefano; Corsaro, Alessandro; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Pino, Albiana; Chiovitti, K.; Paludi, D.; Russo, C.; Sparatore, A.; Aceto, A.; Boido, Vito; Sparatore, Fabio; Florio, Tullio
Epimerization of lupinine to epilupinine and vice versa. Reexamination of the structures of lupinal and epilupinal
2005-01-01 Sparatore, A.; Tasso, Bruno; Boido, Vito; Sparatore, Fabio
Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction
2018-01-01 Tonelli, Michele; Cichero, Elena; Mokhtar Mahmoud, Alì; Rabbito, Alessandro; Tasso, Bruno; Fossa, Paola; Ligresti, Alessia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(+)-Laburnamine, a natural selective ligand and partial agonist for the α4β2 nicotinic receptor subtype | 1-gen-2013 | Tasso, Bruno; Novelli, Federica; Sparatore, Fabio; F., Casoli; C., Gotti | |
Acridine derivatives as anti-BVDV agents | 1-gen-2011 | Tonelli, Michele; Vettoretti, G; Tasso, Bruno; Novelli, Federica; Boido, Vito; Sparatore, Fabio; Busonera, B; Ouhtit, A; Farci, P; Blois, S; Giliberti, G; La Colla, P. | |
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines | 1-gen-2014 | Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Anna, Sparatore; Boido, Vito; Sparatore, Fabio; Sara, Cannas; Paola, Molicotti; Stefania, Zanetti; Silvia, Parapini; Roberta, Loddo | |
Antiviral activity of benzimidazole derivatives. II Antiviral activity of 2-phenylbenzimidazole derivatives. | 1-gen-2010 | Tonelli, Michele; Simone, M; Tasso, Bruno; Novelli, Federica; Boido, Vito; Sparatore, Fabio; Paglietti, G; Pricl, S; Gilberti, G; Blois, S; Ibba, C; Sanna, G; Loddo, R; LA COLLA, P. | |
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents | 1-gen-2014 | Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Vazzana, Iana; Sparatore, Anna; Boido, Vito; Sparatore, Fabio; La Colla, Paolo; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, Bernardetta; Farci, Pamela; Ibba, Cristina; Loddo, Roberta | |
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5 | 1-gen-2015 | Roberta, Loddo; Novelli, Federica; Anna, Sparatore; Tasso, Bruno; Tonelli, Michele; Boido, Vito; Sparatore, Fabio; Gabriella, Collu; Ilenia, Delogu; Gabriele, Giliberti; Paolo, La Colla | |
Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives | 1-gen-2009 | Tonelli, Michele; Vazzana, Iana; Tasso, Bruno; Boido, Vito; Sparatore, Fabio; Fermeglia, M.; Paneni, M. S.; Posocco, P.; Pricl, S.; LA COLLA, P.; Ibba, C.; Secci, B.; Collu, G.; Loddo, R. | |
Benzimidazole derivatives endowed with potent antileishmanial activity | 1-gen-2018 | Tonelli, Michele; Gabriele, Elena; Piazza, Francesca; Basilico, Nicoletta; Parapini, Silvia; Tasso, Bruno; Loddo, Roberta; Sparatore, Fabio; Sparatore, Anna | |
Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles | 1-gen-2017 | Cichero, Elena; Tonelli, Michele; Novelli, Federica; Tasso, Bruno; Delogu, I; Loddo, R.; Bruno, Olga; Fossa, Paola | |
BMI-1 inhibition fights cancer chemoresistance by altering redox homeostasis and inducing lipid peroxidation | 1-gen-2023 | Valenti, Ge; Tasso, B; Traverso, N; Monteleone, L; Marengo, B; Domenicotti, C | |
Btk inhibitors: a medicinal chemistry and drug delivery perspective | 1-gen-2021 | Brullo, C.; Villa, C.; Tasso, B.; Russo, E.; Spallarossa, A. | |
CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation | 1-gen-2013 | M., Sala; D., Braida; L., Pucci; I., Manfredi; M. J., Marks; C. R., Wageman; S. R., Grady; B., Loi; S., Fucile; F., Fasoli; M., Zoli; Tasso, Bruno; Sparatore, Fabio; F., Clementi; C., Gotti | |
Celecoxib Inhibits Prion Protein 90-231-Mediated Pro-inflammatory Responses in Microglial Cells | 1-gen-2016 | Villa, Valentina; THELLUNG DE COURTELARY, Stefano; Corsaro, Alessandro; Novelli, Federica; Tasso, Bruno; Colucci D’Amato, L.; Gatta, Elena; Tonelli, Michele; Florio, Tullio | |
Cytisine derivatives as ligands for neuronal nicotine receptors and with various pharmacological activities | 1-gen-2003 | Canu, Caterina; Tasso, Bruno; Boido, Vito; Sparatore, Fabio | |
Differential modulation of SIRT6 deacetylase and deacylase activities by lysine-based small molecules | 1-gen-2020 | Sociali, G.; Liessi, N.; Grozio, A.; Caffa, I.; Parenti, M. D.; Ravera, S.; Tasso, B.; Benzi, A.; Nencioni, A.; Del Rio, A.; Robina, I.; Millo, E.; Bruzzone, S. | |
Discovery of Novel Thiazole-Based SIRT2 Inhibitors as Anticancer Agents: Molecular Modeling, Chemical Synthesis and Biological Assays | 1-gen-2024 | Piacente, F.; Guccione, G.; Scarano, N.; Lunaccio, D.; Miro, C.; Abbotto, E.; Salis, A.; Tasso, B.; Dentice, M.; Bruzzone, S.; Cichero, E.; Millo, E. | |
Discovery of novel VX-809 hybrid derivatives as F508del-CFTR correctors by molecular modeling, chemical synthesis and biological assays | 1-gen-2020 | Parodi, A.; Righetti, G.; Pesce, E.; Salis, A.; Tasso, B.; Urbinati, C.; Tomati, V.; Damonte, G.; Rusnati, M.; Pedemonte, N.; Cichero, E.; Millo, E. | |
Efficacy of novel acridine derivatives in the inhibition of hPrP90-231 prion protein fragment toxicity | 1-gen-2011 | Villa, Valentina; Tonelli, Michele; THELLUNG DE COURTELARY, Stefano; Corsaro, Alessandro; Tasso, Bruno; Novelli, Federica; Canu, Caterina; Pino, Albiana; Chiovitti, K.; Paludi, D.; Russo, C.; Sparatore, A.; Aceto, A.; Boido, Vito; Sparatore, Fabio; Florio, Tullio | |
Epimerization of lupinine to epilupinine and vice versa. Reexamination of the structures of lupinal and epilupinal | 1-gen-2005 | Sparatore, A.; Tasso, Bruno; Boido, Vito; Sparatore, Fabio | |
Exploring the effectiveness of novel benzimidazoles as CB2 ligands: synthesis, biological evaluation, molecular docking studies and ADMET prediction | 1-gen-2018 | Tonelli, Michele; Cichero, Elena; Mokhtar Mahmoud, Alì; Rabbito, Alessandro; Tasso, Bruno; Fossa, Paola; Ligresti, Alessia |