Sfoglia per Titolo
1,5-Benzodiazepines. Part XIII. Substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines and 4H-imidazo[1,2-a][1,5]benzodiazepin-5-amines as analgesic, anti-inflammatory and/or antipyretic agents with low acute toxicity
2002-01-01 Grossi, Giancarlo; DI BRACCIO, Mario; Roma, Giorgio; V., Ballabeni; M., Tognolini; F., Calcina; E., Barocelli
[1,5-benzodiazepines. V. Synthesis of pyrazolo (3,4-b)(1,5)benzodiazepines and 5H-pyrimido(4,5-b)(1,5)benzodiazepines].
1983-01-01 Roma, G; Balbi, Alessandro; Ermili, A; Vigevani, E.
1,5-Benzodiazepines. X. Dialkylamino substituted 1,5-benzodiazepine and [1,2,4]triazolo[4,3-a][1,5]benzodiazepine derivatives with inhibitory activity on PAF-induced platelet aggregation
1992-01-01 Mario Di, Braccio; Giorgio, Roma; Grossi, Giancarlo; Giuliana, Leoncini; Mitzi, Maresca
1,6 Naphthyridines repurposing: from antiproliferative to antiviral
2018-01-01 Frasson, I.; Spanò, V.; Carbone, A.; Richter, S. N.; Barraja, P.; Montalbano, A.
1,8-Naphthyridines II. 2,4-Disubstituted N,N-dialkyl-1,8-naphthyridine-3-carboxamides with anti-inflammatory and/or antiaggressive activities
1994-01-01 DI BRACCIO, Mario; Roma, Giorgio; Ghia, M.; Mattioli, Francesca
1,8-Naphthyridines III. N,N-Dialkyl-5-chloro[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides with anti-inflammatory activity
1997-01-01 DI BRACCIO, Mario; Roma, Giorgio; Grossi, Giancarlo; Ghia, M.; Mattioli, Francesca
1,8-Naphthyridines IV. 9-substituted N,N-dialkyl-5-(alkylamino or cycloalkylamino) [1,2,4]triazolo[4,3-a][1, 8]naphthyridine-6-carboxamides, new compounds with anti-aggressive and potent anti-inflammatory activities
2000-01-01 Roma, Giorgio; DI BRACCIO, Mario; Grossi, Giancarlo; Mattioli, Francesca; Ghia, M.
1,8-Naphthyridines IX. Potent anti-inflammatory and/or analgesic activity of a new group of substituted 5-amino[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides, of some their Mannich base derivatives and of one novel substituted 5-amino-10-oxo-10Hpyrimido[ 1,2-a][1,8]naphthyridine-6-carboxamide derivative
2014-01-01 Mario Di Braccio, A; Grossi, Giancarlo; Alfei, Silvana; Vigilio Ballabeni, C; Massimiliano Tognolini, C; Lisa Flammini, C; Carmine Giorgio, C; Simona Bertoni, C; Elisabetta Barocelli, C.
1,8-Naphthyridines V.Novel N-substituted 5-amino-N,N-diethyl-9-isopropyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, as potent anti-inflammatory and/or analgesic agents completely devoid of acute gastrolesivity
2005-01-01 Grossi, Giancarlo; DI BRACCIO, Mario; Roma, Giorgio; Ballabeni, V.; Tognolini, M.; Barocelli, E.
1,8-Naphthyridines VI. Synthesis and anti-inflammatory activity of 5-(alkylamino)-N,N-diethyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6 carboxamides with a new substitution pattern on the triazole ring
2008-01-01 DI BRACCIO, Mario; Grossi, Giancarlo; Roma, Giorgio; D., Piras; Mattioli, Francesca; Gosmar, Marzia
1,8-Naphthyridines VII. New substituted 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides and their isosteric analogues, exhibiting notable anti-inflammatory and/or analgesic activities, but no acute gastrolesivity
2008-01-01 Roma, Giorgio; Grossi, Giancarlo; DI BRACCIO, Mario; Piras, D.; Ballabeni, V.; Tognolini, M.; Bertoni, S.; Barocelli, E.
1,8-Naphthyridines VIII. Novel 5-aminoimidazo[1,2-a][1,8]naphthyridine-6-carboxamide and 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamide derivatives showing potent analgesic or anti-inflammatory activity, respectively, and completely devoid of acute gastrolesivity.
2010-01-01 Giorgio, Roma; DI BRACCIO, Mario; Grossi, Giancarlo; Daniela, Piras; Vigilio, Ballabeni; Massimiliano, Tognolini; Simona, Bertoni; Elisabetta, Barocelli
1-(Arylalkyl)quinolizidine derivatives and thio-isosteric analogues as ligands for sigma receptors
2004-01-01 A., Sparatore; Novelli, Federica; Sparatore, Fabio
(1-3)-β-d-glucan in cerebrospinal fluid is useful for the diagnosis of central nervous system fungal infections.
2013-01-01 Mikulska, MALGORZATA KAROLINA; Furfaro, Elisa; Del Bono, V; Raiola, Am; Di Grazia, C; Bacigalupo, A; Viscoli, Claudio
The (1-63) region of the p53 transactivation domain aggregates in vitro into cytotoxic amyloid assemblies
2008-01-01 S., Rigacci; M., Bucciantini; Relini, Annalisa; Pesce, Alessandra; Gliozzi, Alessandra; A., Berti; M., Stefani
1-Acyl-, 3-acyl- and 1,3-diacyl-3-furfuryl-1-phenylthioureas with platelet antiaggregating and other activities.
1991-01-01 Ranise, Angelo; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Donnoli, D; Parrillo, C; Cenicola, Ml; Rossi, F.
1-D Convolutional Neural Networks for Touch Modalities Classification
2021-01-01 Gianoglio, C.; Ragusa, E.; Zunino, R.; Valle, M.
1-Hz repetitive TMS over ipsilateral motor cortex influences the performance of sequential finger movements of different complexity
2008-01-01 Avanzino, Laura; Bove, Marco; Trompetto, Carlo; Tacchino, A; Ogliastro, Carla; Abbruzzese, Giovanni
1-Methyl and 1-(2-hydroxyalkyl)-5-(3-alkyl/cycloalkyl/phenyl/naphthylureido)-1H-pyrazole-4-carboxylic acid ethyl esters as potent human neutrophil chemotaxis inhibitors
2009-01-01 Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Schenone, Silvia; Spisani, S; Falzarano, Ms; Varani, K; Barocelli, E; Ballabeni, V; Giorgio, C; Tognolini, M.
1-Phenyl-1H-Indazole derivatives with analgesic and anti-inflammatory activities.
1992-01-01 Mosti, Luisa; L., Sansebastiano; Fossa, Paola; P., Schenone; Mattioli, Francesca
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