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Discovery of novel VX-809 hybrid derivatives as F508del-CFTR correctors by molecular modeling, chemical synthesis and biological assays
2020-01-01 Parodi, A.; Righetti, G.; Pesce, E.; Salis, A.; Tasso, B.; Urbinati, C.; Tomati, V.; Damonte, G.; Rusnati, M.; Pedemonte, N.; Cichero, E.; Millo, E.
Probing Allosteric Hsp70 Inhibitors by Molecular Modelling Studies to Expedite the Development of Novel Combined F508del CFTR Modulators
2021-01-01 Sabbadini, Roberto; Pesce, Emanuela; Parodi, Alice; Mustorgi, Eleonora; Bruzzone, Santina; Pedemonte, Nicoletta; Casale, Monica; Millo, Enrico; Cichero, Elena
Nbd2 is required for the rescue of mutant f508del cftr by a thiazole-based molecule: A class ii corrector for the multi-drug therapy of cystic fibrosis
2021-01-01 Brandas, C.; Ludovico, A.; Parodi, A.; Moran, O.; Millo, E.; Cichero, E.; Baroni, D.
Journey on VX-809-Based Hybrid Derivatives towards Drug-like F508del-CFTR Correctors: From Molecular Modeling to Chemical Synthesis and Biological Assays
2022-01-01 Parodi, Alice; Righetti, Giada; Pesce, Emanuela; Salis, Annalisa; Tomati, Valeria; Pastorino, Cristina; Tasso, Bruno; Benvenuti, Mirko; Damonte, Gianluca; Pedemonte, Nicoletta; Cichero, Elena; Millo, Enrico
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Discovery of novel VX-809 hybrid derivatives as F508del-CFTR correctors by molecular modeling, chemical synthesis and biological assays | 1-gen-2020 | Parodi, A.; Righetti, G.; Pesce, E.; Salis, A.; Tasso, B.; Urbinati, C.; Tomati, V.; Damonte, G.; Rusnati, M.; Pedemonte, N.; Cichero, E.; Millo, E. | |
Probing Allosteric Hsp70 Inhibitors by Molecular Modelling Studies to Expedite the Development of Novel Combined F508del CFTR Modulators | 1-gen-2021 | Sabbadini, Roberto; Pesce, Emanuela; Parodi, Alice; Mustorgi, Eleonora; Bruzzone, Santina; Pedemonte, Nicoletta; Casale, Monica; Millo, Enrico; Cichero, Elena | |
Nbd2 is required for the rescue of mutant f508del cftr by a thiazole-based molecule: A class ii corrector for the multi-drug therapy of cystic fibrosis | 1-gen-2021 | Brandas, C.; Ludovico, A.; Parodi, A.; Moran, O.; Millo, E.; Cichero, E.; Baroni, D. | |
Journey on VX-809-Based Hybrid Derivatives towards Drug-like F508del-CFTR Correctors: From Molecular Modeling to Chemical Synthesis and Biological Assays | 1-gen-2022 | Parodi, Alice; Righetti, Giada; Pesce, Emanuela; Salis, Annalisa; Tomati, Valeria; Pastorino, Cristina; Tasso, Bruno; Benvenuti, Mirko; Damonte, Gianluca; Pedemonte, Nicoletta; Cichero, Elena; Millo, Enrico |
Mostrati risultati da 1 a 4 di 4
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